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3-({1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}methyl)-4-methoxyphenol
2-fluoro-N-{[8-(3-methylfuran-2-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
methyl (2S)-1-[(4-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]pyrrolidine-2-carboxylate
1-[3-(morpholin-4-yl)piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
1-[2-(cyclohexylmethyl)morpholin-4-yl]-3-(1,2-oxazolidin-2-yl)propan-1-one
1-ethyl-4-({4-oxo-3H,4H-thieno[2,3-d]pyrimidin-3-yl}methyl)pyrrolidin-2-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
1-ethyl-2-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-imidazol-2-yl)-1H-imidazole
6-(cyclopropylmethoxy)-1-(pyridin-3-ylmethyl)-4-(2,2,3,3-tetramethylcyclopropanecarbonyl)-1,4-diazepan-2-one
3-(3,4-difluorophenyl)-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-(2-phenylethyl)-3-(pyrazin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-6-(pyridine-3-sulfonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)piperidin-4-amine
N-[2-(dimethylamino)ethyl]-7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
8-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
ethyl 5-[2-(7-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-{4-[1-(4-phenylbutyl)-1H-imidazol-2-yl]-1H-1,2,3-triazol-1-yl}piperidine
5-ethyl-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidin-2-amine
8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(2-methylpropyl)benzoyl]-4-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
2-[2-(morpholin-4-ylmethyl)-4-(pyrazin-2-yl)phenoxy]-1-(4-phenylazepan-1-yl)ethan-1-one
[1-methyl-5-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
(2R,3S,6R)-5-(5-fluoro-2-methylbenzoyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
4-fluoro-N-(2-{[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidin-3-yl]formamido}ethyl)benzamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]propanamide
2-(2-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}phenoxy)ethan-1-ol
3-(2-methylpropyl)-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazole
2-(2,4-dioxoimidazolidin-1-yl)-N-[3-(1H-indazol-1-yl)propyl]acetamide
(1S,9R)-11-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
(2S,4R)-1-(2-amino-6-methylpyrimidin-4-yl)-N-methyl-4-[2-(5-methyl-1H-pyrazol-1-yl)acetamido]pyrrolidine-2-carboxamide
1-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(4-methylphenyl)propan-1-one
(2S,4S)-4-[(4-methoxyphenyl)sulfanyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-1-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
1-{2,7-diazaspiro[4.5]decan-2-yl}-3-(3,4-dimethylphenyl)propan-1-one
[(3-methoxyphenyl)methyl](prop-2-en-1-yl){[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amine
2-cyclohexyl-N-(pyrimidin-4-ylmethyl)-1,3-benzoxazole-6-carboxamide
N-methyl-4-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
N-[(2,4-dimethylphenyl)(pyridin-3-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-(4-fluorophenoxymethyl)-1-(2-methyl-1,3-thiazole-5-carbonyl)piperidine
methyl[(2-phenyl-1,3-oxazol-4-yl)methyl]{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-[4-(4-fluorophenyl)-2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy]-N-[(2-methoxyphenyl)methyl]acetamide
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
N-ethyl-2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(oxolan-2-ylmethyl)acetamide
N-(propan-2-yl)-1-{1-[5-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
N-[(2R,3R)-2-ethoxy-1'-(1H-pyrazol-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
1-(1-benzylpiperidin-4-yl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(quinoxaline-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one