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8-[(3,5-dichloropyridin-4-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-[3-(propan-2-yloxy)benzoyl]piperidine
3-(2-{4-azatricyclo[4.3.1.13,8]undecan-4-yl}-2-oxoethyl)-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
(3aR,6aS)-5-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(2,5-difluorophenyl)cyclopropyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(2,3-dimethylphenyl)-4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
5-chloro-N-cyclohexyl-3-methyl-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-4-[(4-fluorophenyl)methyl]piperazin-2-one
methyl 3-(2-methoxyacetamido)-5-[(naphthalen-1-ylformamido)methyl]benzoate
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
1-(2-phenoxyethyl)-4-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
3-(oxolan-2-yl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}propan-1-one
methyl 4-[5-methyl-4-({2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}methyl)-1,3-oxazol-2-yl]benzoate
(5-{[(butan-2-yl)(3-phenylprop-2-yn-1-yl)amino]methyl}furan-2-yl)methanol
N-(2-methoxyethyl)-1-(3-methylbutyl)-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{[(1R,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinolin-4-ol
4-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]pyrimidine
methyl 3-[(2,5-dimethylphenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[4-(3,5-difluoropyridine-2-carbonyl)-1,4-oxazepan-6-yl]methanol
N-cyclopentyl-1-(2-methylpropyl)-5-[2-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]pyrazin-2-ol
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-(pyridin-3-yl)ethan-1-one
3-{[benzyl(methyl)amino]methyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-(2-ethoxyethyl)-2-oxo-N-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-(1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-ethyloxane-4-carboxamide
N-({7-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
1-(1H-imidazol-2-ylmethyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
ethyl 2-(1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
5-oxo-1-(propan-2-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}pyrrolidine-3-carboxamide
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
(1R,3S)-3-(2-aminoethoxy)-7-[2-(dimethylamino)benzoyl]-7-azaspiro[3.5]nonan-1-ol
ethyl 1-benzyl-5-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[(3-chlorophenyl)methyl]-N-[1-(1H-indol-1-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
4-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-6-methylpyrimidin-2-amine
5-chloro-4,6-dimethyl-2-[4-(2-phenylethyl)piperazin-1-yl]pyridine-3-carbonitrile
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[1-(pyrazin-2-yl)piperidin-3-yl]acetamide
1-[3-(4-tert-butylphenoxy)-2-hydroxypropyl]-3-(1,3-dihydro-2-benzofuran-5-yl)urea
3-[(2R,3R,6R)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[(2R,3R)-1'-(3-methylthiophene-2-carbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
7-[(3-methoxyphenyl)methyl]-2-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
N-(4-chloro-3-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazine-1-carbonyl}phenyl)acetamide
1-{1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
6-(2-chlorobenzoyl)-N-[3-(2-oxoimidazolidin-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-7-oxo-N-[2-(thiophen-2-yl)ethyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-3-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)urea
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-3-yl)acetamide
2-(3-fluorophenoxymethyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide