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1-[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]-2-(pyridin-4-yl)ethan-1-one
methyl (2S)-1-[2-(4-benzamido-1H-pyrazol-1-yl)acetyl]pyrrolidine-2-carboxylate
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)benzamide
2-fluoro-5-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
6-[3-(4-methoxy-2-methylbenzoyl)piperidine-1-carbonyl]-1H-indole
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
[(3R,4R)-1-(4-cyclopentylpyrimidin-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
2-(1H-indazol-3-yl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)acetamide
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-(2-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
N-cyclopropyl-3-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}propanamide
2-{4-[5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}phenol
5-({4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptane-2-carbonyl]-1,3-oxazol-2-yl}methoxy)-2-methyl-1,3-benzothiazole
3-{2-[2-(cyclopropylmethyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}imidazolidine-2,4-dione
(3S,4R)-4-methyl-1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]piperidine-3,4-diol
methyl 7-oxo-9-(3-phenylpropoxy)-3-[2-(piperidin-1-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methyl-6-(2-methylpropyl)pyrimidine-4-carboxamide
5-{[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)-4-hydroxybenzamide
(3aS,6aR)-5-[(2,6-difluorophenyl)methyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-{3-[3-(2-phenylethyl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
N-methyl-N-(1,3-thiazol-4-ylmethyl)-6-[(2,4,5-trimethoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3-[2-(2,6-difluorophenyl)ethyl]piperidine
3-amino-1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}pyrrolidine-3-carboxylic acid
(3S,4R)-1-[2-(2-ethoxyphenoxy)ethyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
6-(methoxymethyl)-N-methyl-N-(piperidin-4-yl)pyridine-2-carboxamide
2-(2,6-dimethoxy-4-methylphenyl)-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
2-(2-{5-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrrol-1-yl)pyrimidine
4-[(dipropylamino)methyl]-N-ethyl-N-(pyridin-2-ylmethyl)benzamide
1-(cyclopropylmethyl)-5-[3-(2-methoxyphenyl)propanoyl]-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-methyl-N-(2-methylpropyl)-5,6-dihydro-1,4-dioxine-2-carboxamide
(1R,3S)-3-methoxy-7-(1-phenylcyclohexanecarbonyl)-7-azaspiro[3.5]nonan-1-ol
N-[(2,3,4-trimethoxyphenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
4-({[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]amino}methyl)phenol
(4S)-4-acetamido-5-oxo-5-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}pentanamide
(2E)-1-[(3R,4R)-3-hydroxy-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-1-yl]-3-phenylprop-2-en-1-one
1,3-dimethyl-6-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,9aR)-8-(naphthalene-1-carbonyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-(cyclopropylmethoxy)-1-(pyridin-3-ylmethyl)-4-[4-(thiophen-2-yl)butanoyl]-1,4-diazepan-2-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-3-(pyrazin-2-yl)propanamide
N-(1-{7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylbenzamide
5-{1-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}-2-(pyridin-2-yl)pyrimidine
4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-1-(2-methoxyphenyl)-5-methylpiperazin-2-one
N-(isoquinolin-5-ylmethyl)-N-methyl-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
1-{5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}azetidin-3-ol
4-[2-(1H-pyrazol-1-yl)ethyl]-1-(1,3-thiazol-4-ylmethyl)piperidine
7-(2-methoxyphenyl)-2-(3-propyl-1,2-oxazol-5-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]pyridin-1-ium-1-olate
9-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
methyl (2S,4S)-4-(2,3-dimethyl-1H-indole-7-amido)-1-[(2-fluorophenyl)methyl]pyrrolidine-2-carboxylate