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8-(6-methoxypyridin-3-yl)quinolin-4-amine
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-fluorobenzamide
N-[2-(ethanesulfonyl)ethyl]-4-methylpyrimidine-5-carboxamide
6-[3-(4-methylphenyl)propanoyl]-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[(5-phenylthiophen-2-yl)methyl]piperidin-4-ol
1-[(4-chlorophenyl)methyl]-4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
4-{[6-(6-methoxypyridin-3-yl)pyridin-3-yl]methyl}morpholine
3-[3-methyl-1-(2-methylphenyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]benzonitrile
N1-(1,4-dithiepan-6-yl)-N2-(3-methylpyridin-2-yl)ethane-1,2-diamine
4-(2-{1-[2-(4-fluorophenoxy)ethyl]piperidin-2-yl}ethyl)morpholine
ethyl 1-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(ethoxycarbonyl)-1H-pyrazol-5-yl]methyl}piperidine-4-carboxylate
(1S,4S)-2-(3-chloro-4-methoxyphenyl)-5-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
[5-methyl-7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
6-[2-({[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido}methyl)-2,3-dihydro-1-benzofuran-7-yl]pyridine-3-carboxamide
2-{3-[4-(1-ethoxyethyl)phenyl]phenoxy}acetamide
N-(2,2-dimethyloxan-4-yl)-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
3-(4-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)propanamide
methyl (1S,3S,3aR,6aS)-5-ethyl-4,6-dioxo-1-phenyl-3-(pyridin-3-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(2S)-N-[2-(3,5-dimethylphenoxy)ethyl]-2-acetamido-N-methylpentanediamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]propan-1-one
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-{[(4-fluorophenyl)methyl]amino}benzamide
5-[(2-methoxyethyl)(methyl)amino]-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
9-[(5-ethylfuran-2-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2,2-dimethyloxan-4-yl)-1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1'-(quinoxaline-5-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
(3aR,6aR)-2-cyclopropanecarbonyl-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-{4-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
5-chloro-N-(cyclobutylmethyl)-4,6-dimethyl-2-oxo-N-(oxolan-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
3-cyano-N-[1-(1-methyl-1H-imidazol-2-yl)butyl]benzamide
1-(2,6-difluoro-3-methylbenzoyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[3-(pyridin-3-yl)propyl]pyrrolidin-3-yl]acetamide
4,4-difluoro-N-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}piperidine-1-carboxamide
1-{3-[({[4-(methylsulfanyl)phenyl]methyl}amino)methyl]phenoxy}-3-(morpholin-4-yl)propan-2-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N,2,3-trimethylquinoxaline-6-carboxamide
1-(cyclobutylmethyl)-3-hydroxy-3-({4-[(pyrimidin-2-yl)amino]piperidin-1-yl}methyl)piperidin-2-one
2-[2-(4-methoxybenzoyl)-1H-imidazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-4-{5-[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]furan-2-yl}but-3-yn-2-ol
1-benzyl-4-(2,5-dimethoxybenzoyl)-6-methoxy-1,4-diazepan-2-one
2-[2-(2-phenylmorpholin-4-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-[(3-fluorophenyl)methyl]piperidin-4-yl]methanol
(1S,5R)-6-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
7-(1-benzofuran-2-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
(1S,5R)-3-benzyl-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(3-methoxyphenyl)methyl]-4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-2-one
4-(2-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}-2-methylpropyl)morpholine
2-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
(1S,5R)-6-benzyl-3-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane