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N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1,3-benzothiazole-6-carboxamide
1-[1-(2-cyclopropylacetyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
6-[(4-fluorophenyl)methoxy]-1-(propan-2-yl)-4-[4-(1H-pyrazol-1-yl)benzoyl]-1,4-diazepan-2-one
(2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
3-methyl-1-(1-{6-[(1-methylpiperidin-4-yl)amino]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
2-{4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
2-(pyrimidin-2-ylsulfanyl)-N-{[5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2-{1-[2-(1H-indol-3-yl)ethyl]-1H-1,2,3-triazol-4-yl}benzoic acid
2-(dimethylamino)-N,4-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidine-5-carboxamide
5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]-N-methylpyrimidin-2-amine
N-{[2-(4-cyclobutaneamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
N-ethyl-5-{1-[(4-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}pyrimidin-2-amine
benzyl N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
(4aR,7aS)-1-(cyclopropylmethyl)-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-ethyl-6-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
1-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
6-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexan-1-ol
N-[1-(7-{[4-(dimethylamino)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-3-phenylpropanamide
1-ethyl-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,3,5-trimethyl-1H-pyrazole-4-carboxamide
1-{3-methoxy-5-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}-1H-1,2,3,4-tetrazole
(3aS,6aS)-1-[3-(benzyloxy)propyl]-octahydropyrrolo[2,3-c]pyrrole
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(5-methyl-1,2-oxazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aS,8aR)-6-(cyclopropylmethyl)-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-cyclopropyl-3-{1-[2-(2-methylphenyl)acetyl]piperidin-4-yl}propanamide
4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-1,2-dihydroisoquinolin-1-one
5-(azepane-1-carbonyl)-N-benzyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]benzamide
N,1-dimethyl-N-[(3-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperidin-4-amine
4-hydroxy-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
ethyl 2-[(5-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}pyrimidin-2-yl)amino]acetate
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-cyclohexyl-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-(prop-2-yn-1-yl)propanamide
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4,4,4-trifluorobutan-1-one
1-(4-chloro-1-methyl-1H-indole-2-carbonyl)-4-(hydroxymethyl)piperidin-4-ol
N-[4-methoxy-3-(4H-1,2,4-triazol-4-yl)phenyl]acetamide
3-(3-methylbut-2-en-1-yl)-1-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]piperidine-3-carboxylic acid
N,1-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-[2-(4-fluorophenyl)ethyl]-4-{4-[2-(4-methylphenoxy)acetyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-(3-fluoro-4-methoxybenzoyl)piperidine
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-2-methyl-1,3-thiazole-4-carboxamide
2-(2-ethylphenyl)-2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}acetic acid
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(phenylsulfanyl)ethan-1-one
2-{1-[2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl}-5-methyl-1H-1,3-benzodiazole
N-[2-(2-ethylphenoxy)ethyl]-N,7-dimethylpyrazolo[1,5-a]pyrimidine-6-carboxamide
4-[(5-methoxy-1H-indazol-3-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
2-[(3aS,6aS)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-octahydropyrrolo[3,4-b]pyrrol-5-yl]-1,3-thiazole-4-carboxamide
1-(7-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-(thiophen-2-yl)propan-1-one
4-(2,5-dichlorophenyl)-2-methylpyrimidine
(3S,4S)-1-(2-fluoro-5-sulfamoylbenzoyl)-4-propylpyrrolidine-3-carboxylic acid