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2-[(1S,5R)-3-[(2-chlorophenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)methyl]-1,2-dihydroquinoxalin-2-one
methyl({[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl})(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
3-{5-[2-(dimethylamino)phenyl]-3-methyl-1H-1,2,4-triazol-1-yl}-4-fluorobenzene-1-sulfonamide
2-(1H-1,3-benzodiazol-1-yl)-1-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]propan-1-one
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-3-(2-oxopyrrolidin-1-yl)benzamide
4-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}-1,4-oxazepan-6-ol
4-methyl-7-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)-2H-chromen-2-one
N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(thiophen-2-yl)acetamide
5-[1-(4-fluorophenyl)cyclopropyl]-3-(2-methoxyethyl)-1,2,4-oxadiazole
1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,3-benzodiazole
methyl({[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl})(pyrazin-2-ylmethyl)amine
2-cyclopropyl-N-(furan-2-ylmethyl)-4-methyl-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
2-(4-chlorophenoxy)-1-(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)ethan-1-one
N-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
1-(2,3-difluorophenyl)-3-[(1R,2S)-2-(methoxymethyl)cyclopentyl]urea
N-(furan-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]-N-(prop-2-yn-1-yl)-1,2-oxazole-5-carboxamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
[2-(azepan-1-yl)ethyl](ethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}furan-2-carboxamide
5-{1-[2-(2-chloro-6-fluorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-[(2-ethoxypyridin-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
8-(adamantan-2-yl)-3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-acetyl-3-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-[(2R,3R)-2-hydroxy-1'-(3-phenylpropyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
3-{1-[(3S,4S)-4-hydroxy-1-(propan-2-yl)pyrrolidin-3-yl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
2-(morpholin-4-yl)-1-{4-[3-(1H-pyrazol-3-yl)phenyl]phenyl}ethan-1-ol
5-{[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-2-methylpyrimidine
methyl({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)(1,3-thiazol-4-ylmethyl)amine
4-[(3-methoxyphenyl)methyl]-3-oxo-N-[3-(propan-2-yl)phenyl]piperazine-1-carboxamide
5-(2-chlorophenyl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methylfuran-2-carboxamide
2-{[2-(hydroxymethyl)piperidin-1-yl]methyl}-4-(pyrazin-2-yl)phenol
3-({[2-(dimethylamino)-6-ethylpyrimidin-4-yl]amino}methyl)-N,N-dimethylbenzamide
4-({[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)-1-methylpiperidin-4-ol
2-{2-[(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)amino]ethyl}-1,2-dihydrophthalazin-1-one
2-(2-{[methyl(2-phenylethyl)amino]methyl}phenyl)-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
N-[(3S,4R)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
5-(1H-1,2,3-benzotriazole-5-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{4-[4-(2-hydroxyethyl)piperidin-1-yl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
7-hydroxy-6-methyl-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1,2,3,4-tetrahydroquinolin-2-one
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-[(4-methylphenyl)methyl]acetamide
1-[2-(7-fluoro-4-oxo-3,4-dihydroquinazolin-3-yl)ethyl]piperidine-3-carboxamide
1-(4-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}thiophen-2-yl)ethan-1-one
methyl 5-{[(2,4-difluorophenyl)methyl]amino}-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(4-fluorophenyl)-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine
3-{1-[2-(pyrrolidin-1-yl)ethyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
[(6-ethoxyquinolin-2-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
(2S)-2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-4-(methylsulfanyl)butan-1-ol