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N-[(2R,3R)-2-methoxy-1'-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
[(3aS,6aS)-2-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
4-({[1-(6-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]amino}methyl)hepta-1,6-dien-4-ol
7-(cyclohexylmethyl)-2-[(4-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
N-{1-[1-(2,4-dimethylbenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,3-dimethylbutanamide
2-{3,5-dimethyl-4-[4-(1,3-oxazol-5-yl)benzenesulfonamido]-1H-pyrazol-1-yl}acetic acid
{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}(methyl)({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)amine
3-[1-(4-cyano-1-methyl-1H-pyrrol-2-yl)-N-(2-phenylethyl)formamido]propanamide
N-(2,4-dimethoxyphenyl)-3-(1-{spiro[2.4]heptane-1-carbonyl}piperidin-4-yl)propanamide
1-(4-{[(benzylsulfamoyl)amino]methyl}piperidin-1-yl)-2-methylpropan-1-one
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]imidazo[1,2-a]pyridine-2-carboxamide
1-(2,2-dimethylcyclopropanecarbonyl)-4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine
1-(3-fluorophenyl)-3-{1-[1-(1H-pyrazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
4-(1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)thiomorpholine
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[3-(propan-2-yloxy)propyl]benzamide
N-[2-(2-fluorophenoxy)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-ethyl-4-[5-(pentan-2-yl)-4-phenyl-1H-imidazol-1-yl]piperidine-1-carboxamide
1-(cyclopropylmethyl)-5-(furan-3-ylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 3-[(3S,4R)-1-[(3-hydroxy-4-methoxyphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
N-(cyclopropylmethyl)-1-[(2-fluorophenyl)methyl]piperidin-3-amine
1-methyl-6-oxo-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1,6-dihydropyridine-3-carboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
5-acetyl-N,2,4-trimethyl-N-[(5-methylfuran-2-yl)methyl]-1H-pyrrole-3-carboxamide
2-(3-{[3-(1H-indol-2-yl)phenyl]carbamoyl}piperidin-1-yl)acetic acid
(3R,5S)-N-[2-(dimethylamino)ethyl]-5-[(4-methylpiperazin-1-yl)methyl]-1-(2-phenylethyl)piperidine-3-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-benzyl-4-[4-(1,4-oxazepan-4-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
(1R,5R)-N,N-dimethyl-6-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(1-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
2-(2,4-dioxo-1,3-thiazolidin-3-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
1-(3,6-dimethylpyrazin-2-yl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylic acid
8-acetyl-2-[(2,6-dimethoxyphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(4-methoxyphenyl)methyl]piperidin-4-ol
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
N-[(5-fluoro-2-methylphenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(2-chlorophenyl)methyl]-2-(2-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-4-phenylphenoxy)acetamide
5-methyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-3-phenyl-1,2-oxazole
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
5-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-[2-(dimethylamino)ethyl]-5-(pyridin-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-{6-chloro-3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2-(furan-2-yl)pyrrolidine
3-benzyl-8-[1-(4-hydroxy-3-methoxyphenyl)propan-2-yl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
[5-({[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amino}methyl)furan-2-yl]methanol
3-[3-({[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,4-dimethylbenzamide
4-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}pyrimidine
3-chloro-6-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide