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1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2-chlorophenyl)ethan-1-one
(1R,5S,6R,7S)-3-(2-aminoethyl)-N-[3-(2-fluorophenyl)propyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]decane-6-carboxamide
1-methyl-4-(5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)-1,4-diazepane
(3S,4S)-4-(4-fluorophenyl)-1-(1H-indol-4-ylmethyl)piperidin-3-ol
2-({5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}(methyl)amino)ethan-1-ol
ethyl 4-[(2-chlorophenyl)methyl]-1-(thiophene-2-carbonyl)piperidine-4-carboxylate
2-(2-fluorophenoxymethyl)-N-(1H-imidazol-2-ylmethyl)-1,3-oxazole-4-carboxamide
2-[6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]pyridine
1-(2-methoxyacetyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
(3S,4S)-1-[3-(3,4-dimethoxyphenyl)propanoyl]-4-propylpyrrolidine-3-carboxylic acid
2-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propane-1,3-diol
3-[2-(dimethylamino)ethyl]-8-(2,6-dimethylhept-5-en-1-yl)-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(5-methylfuran-2-yl)methyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
2-({2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}methyl)-1H-1,3-benzodiazole
methyl 3-{[(3-fluorophenyl)formamido]methyl}-5-(pyridine-4-amido)benzoate
5-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(5-acetamido-2-fluorophenyl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
2-hydroxy-1-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
2-[methyl(pyridin-4-ylmethyl)amino]-1-(3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)ethan-1-one
N-[(1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-3-yl)methyl]acetamide
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}phenoxymethyl)pyridine
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
2-[1-(3-methoxypropyl)pyrrolidin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2E)-N-{[7-(4-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
7-fluoro-2-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3-methyl-1H-indole
3-chloro-4-fluoro-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-benzothiophene-2-carboxamide
N-(1-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-2-phenylethyl)-N-methylthiophene-3-carboxamide
1-[(2-methylphenyl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
2-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1,2-oxazinane
1-[1-(4-methylpent-3-en-1-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-ethyl-3-(3-methoxyphenyl)-N-(oxan-4-ylmethyl)-1H-pyrazole-5-carboxamide
2-(dimethylamino)-N-{[8-(3-phenylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
4-[(2,5-difluorophenyl)methyl]-9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N,3,5-trimethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1H-indole-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy]-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
N-[(6-methylpyridin-2-yl)methyl]-6-[(2-phenyl-1,3-thiazol-5-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-{[7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
2-[5-(1-{[1-(3-methylphenyl)-1H-1,2,3,4-tetrazol-5-yl]sulfanyl}ethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-4-oxo-N-[(3S)-2-oxoazepan-3-yl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-cyclopentyl-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-3-{1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-3-yl}propanamide
2-methyl-4-{3-[2-(1-methyl-1H-pyrazol-3-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
6-chloro-N,N-dimethyl-3-({[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
4-(1H-pyrazol-1-yl)-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
4-{4-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
5-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2-(4H-1,2,4-triazol-4-yl)pyridine
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(1R)-1-phenylethyl]acetamide
5-(4-fluorophenyl)-7-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}pyrazolo[1,5-a]pyrimidine