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1,6-dimethyl-N-[1-(1,3-thiazol-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[1-(5-methoxypyridin-3-yl)-1H-imidazol-2-yl]thiophene-2-carboxylic acid
6-cyclopropyl-N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methylpyrimidin-4-amine
2-cyclobutyl-1-methyl-N-[(4-methylphenyl)methyl]-7-(oxolane-2-amido)-1H-1,3-benzodiazole-5-carboxamide
ethyl(oxan-2-ylmethyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
[4-({methyl[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}methyl)oxan-4-yl]methanol
N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-1,3,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(5-{[(adamantan-2-ylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
(2R,6S)-4-[5-(1H-imidazol-2-yl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]-2,6-dimethylmorpholine
3-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]-1-[2-(morpholin-4-ylmethyl)phenyl]urea
1-ethyl-4-{[methyl({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amino]methyl}pyrrolidin-2-one
1-cyclopropyl-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-(2-methylpropyl)acetamide
N-[2-(4-chlorophenyl)ethyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)acetamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(5-methylthiophen-2-yl)methyl]-decahydro-2,7-naphthyridine-2-sulfonamide
N-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-[2-(2-fluoro-4,5-dimethoxyphenyl)-1H-imidazol-1-yl]-1-phenylethan-1-ol
2-methyl-4-{3-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
N-({8-[(1-acetyl-1H-indol-3-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1-methyl-1H-pyrazole-3-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
6-(3-ethoxyphenyl)-N,N-dimethylpyridine-2-carboxamide
5-methyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N4-cyclopropyl-7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-{4-[1-(pent-2-yn-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}pyridine
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
5,6-dimethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-(trifluoromethyl)pyrimidin-4-amine
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
1-[2-methoxy-6-({methyl[2-(oxan-4-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
2-(4-acetylphenoxy)-1-[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]ethan-1-one
N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)quinoxaline-6-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
3-{5-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
1-(1-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl)-1H-imidazole
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
N,N-dimethyl-3-{[3-(1-methylpiperidin-2-yl)propanamido]methyl}benzamide
6-(2-chlorophenyl)-2-[4-(1,4-diazepan-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
8-(dimethyl-1,2-oxazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(3R,4S)-4-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-1-yl}oxolan-3-ol
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}naphthalene-1-carboxamide
5-(2-chloro-4-fluorophenoxymethyl)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-(2-methoxyphenyl)-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]propanamide
3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1-phenylpyrrolidin-2-one
8-(5-chloropyridine-2-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
N-[(2R,3R)-1'-[(3-hydroxyphenyl)methyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
(5S,9aS,9bS)-5-(1-ethyl-1H-1,3-benzodiazol-2-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one