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N-[2-(5-methylfuran-2-yl)ethyl]-3-[(3-oxopiperazin-1-yl)sulfonyl]benzamide
5-(3-fluorophenoxymethyl)-N-[2-(propan-2-yloxy)ethyl]-1H-pyrazole-3-carboxamide
5-acetyl-6-methyl-3-[2-(2-phenylethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrimidine
methyl 4-[4-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperazin-1-yl]benzoate
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-fluorophenyl)methyl]acetamide
2-(pyridin-3-yl)-5-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrimidine
N-(4-{2-amino-3-cyano-7-hydroxy-5H-indeno[1,2-b]pyridin-4-yl}phenyl)acetamide
(3R,4R)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N,1-dimethylpyrrolidine-3-carboxamide
5-[({[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-({[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](methyl)amino}methyl)-4-methylphenol
3-[(4-methoxypyridin-2-yl)methyl]-5-methyl-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-[(3R,4S)-3-[(2-amino-6-methylpyrimidin-4-yl)amino]-4-propylpyrrolidin-1-yl]-2-(methylsulfanyl)ethan-1-one
{[3-cyclopentyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl](phenyl)methyl}(methyl)amine
2-({3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
4-fluoro-N-[3-(4-{[2-(1,3-thiazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]benzene-1-sulfonamide
N-[2-(1H-pyrazol-1-yl)ethyl]-3-[(1,3-thiazol-2-ylmethyl)sulfamoyl]benzamide
methyl 3-[(2-fluoro-4-methoxyphenyl)methyl]-9-[2-(2-fluorophenyl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S,4R)-4-amino-1-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-4-yl]-N-methylpyrrolidine-2-carboxamide
[4-(5-phenyl-1,3,4-thiadiazol-2-yl)-1,4-oxazepan-6-yl]methanol
1-(4-chlorophenyl)-3-(furan-2-yl)-4-[2-(2-methylpyrrolidin-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1,3-benzothiazol-2-ylmethyl)-4-hydroxy-N-methyl-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
(1S,5R)-6-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
3-({[1-butyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]methyl}(methyl)amino)-1λ6-thiolane-1,1-dione
N,N-dimethyl-5-(1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}pyrrolidin-2-yl)thiophene-2-carboxamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(1-methyl-3-phenyl-1H-pyrazol-5-yl)formamido]acetic acid
1-[(2,4-difluorophenyl)methyl]-4-ethyl-1,4-diazepan-5-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
2-{1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-1H-imidazol-2-yl}quinoline
N-[(2R,3R)-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-(2,5-dimethoxyphenyl)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidine
N-[(3R,4S)-4-cyclopropyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl]methanesulfonamide
N-[3-(1H-indol-2-yl)phenyl]-1-(3-methylbutanoyl)piperidine-4-carboxamide
methyl 4-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-oxobutanoate
ethyl 4-[1-(2-cyclopentylacetyl)piperidin-3-yl]piperazine-1-carboxylate
1-{5-[1-(3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
(3R,5S)-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-1H-1,2,3-benzotriazole-5-carboxamide
N-(4-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}phenyl)ethane-1-sulfonamide
N-{3-[(butan-2-yl)(pyridin-3-ylmethyl)carbamoyl]phenyl}-2-methylfuran-3-carboxamide
N,N-dimethyl-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carboxamide
2-(3-benzyl-1H-1,2,4-triazol-5-yl)-5-methoxy-1H-indole
N-[2-(3,4-dihydro-2H-1-benzopyran-6-ylformamido)ethyl]-2,2,2-trifluoroacetamide
2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-(furan-2-ylmethyl)piperidine
methyl 4-(4-{1-[2-(dimethylamino)-N-methylacetamido]-2-phenylethyl}piperidin-1-yl)-4-oxobutanoate
5-(butoxymethyl)-3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole