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3-(hydroxymethyl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-3-ol
3-(azepane-1-carbonyl)-5-(morpholin-4-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
6-(2,2-dimethyloxan-4-yl)-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
1-[(2-chlorophenyl)methyl]-1-(2-hydroxyethyl)-3-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N-methylacetamide
4-{[4-methyl-5-(1-methylpiperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}morpholine
N-({1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
1-methyl-4-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperazine
(3S,4S)-4-cyclopropyl-1-(3-methylbut-2-enoyl)pyrrolidine-3-carboxylic acid
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
methyl 5-[(2,2-dimethylpropyl)amino]-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(2-phenoxyethyl)-1-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,4-diazepan-5-one
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(1H-imidazol-1-yl)ethan-1-one
1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
(4-{[(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]methyl}oxan-4-yl)methanol
1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenyl-1,4-diazepane
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[(4-methyl-1,3-thiazol-2-yl)methyl]propanamide
1-ethyl-N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-3,5-dimethyl-1H-pyrazole-4-carboxamide
methyl 3-[2-(3-methylphenyl)acetyl]-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-methyl-4-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
3-(2,6-dimethylpyridin-3-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
1-{[(2S,4S)-1-[2-(2,3-dihydro-1H-inden-5-yloxy)-2-methylpropanoyl]-4-fluoropyrrolidin-2-yl]methyl}-3,3-dimethylurea
5-methoxy-N-(2-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)furan-2-carboxamide
2,2,2-trifluoro-N-{2-[(2-methyl-1H-1,3-benzodiazol-4-yl)formamido]ethyl}acetamide
N-{[5-({[(3-ethoxyphenyl)methyl](2-hydroxyethyl)amino}methyl)furan-2-yl]methyl}-N-methylmethanesulfonamide
2-{1-benzyl-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-[(2-ethyl-1,3-thiazol-4-yl)methyl]-7-(3-methoxypropyl)-2,7-diazaspiro[4.5]decan-6-one
1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-4-(3-methylpyridin-4-yl)-1,4-diazepane
(2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{methyl[(5-methyl-1,2-oxazol-3-yl)methyl]carbamoyl}pyrrolidine-2-carboxylic acid
5-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-1,2,4-triazol-3-amine
2-methyl-5-{[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]methyl}-1,3,4-oxadiazole
N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
1-methyl-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
1-(4-ethoxy-2-fluorophenyl)-3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]urea
3-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-N-phenylpropanamide
N-methyl-N-(2-phenyl-1-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}ethyl)-2-(1H-pyrazol-1-yl)acetamide
(2R,6R)-4-[(1-ethyl-1H-pyrazol-3-yl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
ethyl 5-{2-azabicyclo[2.2.1]heptan-2-ylmethyl}-1-(1H-1,3-benzodiazol-2-yl)-1H-pyrazole-4-carboxylate
(1S,5R)-6-benzyl-3-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-({[2-(2-aminoethyl)quinazolin-4-yl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
3-ethyl-6-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-3H-imidazo[4,5-b]pyridin-2-amine
2-(methylamino)-N-{1-phenyl-3,6-diazatricyclo[4.3.1.13,8]undecan-9-yl}pyridine-4-carboxamide
3-(2-oxoimidazolidin-1-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
(3S,4R)-4-phenyl-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidine-3-carboxylic acid