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1-(azocan-1-yl)-3-(2-methoxy-4-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
methyl 2-methyl-2-({5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazol-3-yl}formamido)propanoate
(1R,5R)-6-[(2-fluoro-5-methoxyphenyl)methyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1-(5-propylpyrimidin-4-yl)piperidin-4-amine
3-({[(2-aminopyridin-3-yl)methyl]amino}methyl)-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-8-(3,3,5,5-tetramethylcyclohexyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(6-hydroxypyrimidin-4-yl)methyl]-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
methyl (2S,4R)-1-[(5-methylthiophen-2-yl)methyl]-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
4-[1-benzyl-5-(1,2,5-thiadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
5-{[4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-1,2,3,4-tetrazole
[1-(2H-1,3-benzodioxol-4-ylmethyl)-4-benzylpiperidin-4-yl]methanol
ethyl 1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
1-{2-methoxy-5-[(4-methoxypiperidin-1-yl)methyl]phenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
4-{2-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}phenol
(3R,4S)-4-cyclopropyl-1-(2,6-difluorobenzoyl)pyrrolidin-3-amine
2-[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
6-oxo-N-[2-(2-oxopiperidin-1-yl)ethyl]-1-(2-phenylethyl)piperidine-3-carboxamide
3-(2-fluorophenyl)-1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]propan-1-one
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperidine
2-(1-cyclohexyl-4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
1-cyclopentanecarbonyl-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylic acid
dimethyl[(6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-3-yl)methyl]amine
5-(2-methylphenyl)-2-(pyridin-3-yl)-4-[1-(2,3,6-trifluorobenzoyl)piperidin-4-yl]pyrimidine
2-(3-methylbut-2-en-1-yl)-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
4-[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]pyridin-1-ium-1-olate
2-methyl-N-{[8-(quinolin-7-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1,3-thiazole-4-carboxamide
8-(butan-2-yl)-1-(3-methylbutyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,7aS)-1-{2-[methyl(pyridin-2-ylmethyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(2-fluorophenyl)formamido]-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]propanamide
(3R,4S)-1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3,4-dimethylpiperidin-4-ol
5-benzyl-5-[1-(2-ethylbutanoyl)piperidin-4-yl]-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
2-[1-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)pyrrolidin-2-yl]-1,3-thiazole
ethyl 4-{2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
6-methoxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-3-methyl-1-benzofuran-2-carboxamide
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-2-propoxyacetamide
2,4-dimethyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,3-thiazole-5-carboxamide
8-[1-(2-methoxyphenyl)piperidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
8-(2-ethylpyridine-4-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N2,N2-dimethyl-N4-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
N-{3-[4-(butylamino)piperidin-1-yl]phenyl}-3-(trifluoromethyl)benzamide
methyl 5-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-3-(furan-2-amido)-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[(2-cyclohexylpyrimidin-5-yl)methyl]-1-phenylpiperazin-2-one
1-(4-chloro-3-fluorobenzoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-({3-methyl-7-[(2E)-2-methylbut-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[6-(dimethylamino)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(3-chloro-4-methoxyphenyl)-5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)pyridine
1-[2-methoxy-6-({[2-(pyrazin-2-yl)ethyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
4-(2-ethylbutyl)-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide