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6-ethyl-4-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
8-{[4-(azepane-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-4-(piperidin-1-yl)butanamide
1-benzyl-6-(cyclopropylmethoxy)-4-(3-methylbenzoyl)-1,4-diazepan-2-one
6-[4-(4-fluorophenyl)oxan-4-yl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
3-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
dimethyl({1-[4-(4-phenyl-1H-imidazol-5-yl)phenyl]ethyl})amine
N-(adamantan-1-yl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
N-{1-[3-(piperidin-3-yl)benzoyl]piperidin-4-yl}methanesulfonamide
4-(3-methyl-1H-pyrazol-1-yl)-N-(propan-2-yl)aniline
N-benzyl-3-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-N-methylpropanamide
5,6-dimethyl-N-[2-(oxolan-3-yl)ethyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
1-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
4-[4-(dimethylamino)phenyl]-3-methyl-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-[4-(2-ethoxyphenyl)piperazin-1-yl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
3-(cyclohex-1-en-1-ylmethyl)-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
methyl 7-oxo-3-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]amine
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
7-[cyclohexyl(methoxy)methyl]-4-(2,3-dihydro-1-benzofuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
{1-[(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}methanamine
4-ethyl-5-methyl-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]pyrimidin-2-amine
3,3-dimethyl-1-({5-[(3-phenyl-1H-pyrazol-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
1-tert-butyl-4-[4-(1H-pyrrole-2-carbonyl)piperazine-1-carbonyl]pyrrolidin-2-one
8-(2-propyl-1,3-thiazole-4-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(3-acetyl-1H-indol-1-yl)-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]butanamide
N-ethyl-2-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1,3-thiazole-4-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-ethyl-N-(2-hydroxyethyl)-1,3-oxazole-4-carboxamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1-phenyl-1H-pyrazole-4-carboxamide
3-(2-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-4-(pyridin-3-ylmethyl)piperazin-2-one
3-[4-(4-acetylphenyl)piperazine-1-carbonyl]-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3-ethoxybenzoyl)piperidine
1-ethyl-5-({[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(3S,4R)-1-{2-[4-(hydroxymethyl)phenyl]acetyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
(3S,7S)-5-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-triene-3-carboxylic acid
3-ethyl-4-methyl-N-[3-(4-methylpiperazin-1-yl)butyl]-1H-pyrazole-5-carboxamide
(4aS,8aR)-1-(4-hydroxybutyl)-6-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-methoxy-1-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propan-1-one
1-{[4-(2-aminoethyl)phenyl]methyl}-4-cyclopropanecarbonyl-1,4-diazepan-6-ol
3-{[(2,2-dimethylpropyl)amino]methyl}-3-hydroxy-1-[(3-methylphenyl)methyl]piperidin-2-one
1-[2-methoxy-4-({[(1-methylpiperidin-4-yl)methyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
4-(4-methylpiperazin-1-yl)-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
6-methyl-5-[5-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-2-{spiro[2.3]hexane-1-carbonyl}-1,2,3,4-tetrahydro-2,7-naphthyridine
3-{2-[({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(ethyl)amino]-1-hydroxyethyl}phenol
1-[1-ethyl-5-(naphthalene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-{1-oxa-8-azaspiro[4.5]decan-3-yl}-4-sulfamoylbenzamide
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(2-phenylethyl)piperidine
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(furan-3-ylmethyl)-N-methyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide