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4-(4-ethoxy-3-methylphenyl)-4-oxo-N-[2-(pyrrolidine-1-sulfonyl)ethyl]butanamide
{2-oxo-2-[2-oxo-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]ethyl}urea
methyl 1-benzyl-5-({[4-(methoxycarbonyl)phenyl]methyl}amino)-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(1-tert-butyl-1H-pyrazol-4-yl)-7,8-dimethyl-4-(pyrrolidine-1-carbonyl)quinoline
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
[(2-chlorophenyl)methyl]({[2-(2-methoxyphenoxy)pyridin-3-yl]methyl})amine
1-cyclopropyl-1-[(4-ethylphenyl)methyl]-3-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
6-chloro-N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-1-methyl-1H-indole-2-carboxamide
methyl 2-{[2-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-6-[(4-hydroxyphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
4-[(3,5-dimethoxyphenyl)methyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{5-[2-(benzenesulfonyl)ethyl]-1-phenyl-1H-1,2,4-triazol-3-yl}acetamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[1-(2-methoxyphenyl)ethyl]-N-methyl-1,2-oxazole-3-carboxamide
3-{2,8-diazaspiro[4.5]decan-3-ylformamido}-N-(1,3-thiazol-2-yl)propanamide
2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-propyl-1,3,4-oxadiazole
(2S,4R)-N,1-dimethyl-4-{4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanamido}pyrrolidine-2-carboxamide
6-fluoro-4-[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydroquinolin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
1-(difluoromethyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]thiophene-3-carboxamide
2-{5-[2-(ethylamino)pyrimidin-5-yl]-3-(4-fluorophenoxymethyl)-1H-1,2,4-triazol-1-yl}acetic acid
[(2-methoxyphenyl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
4-(dimethyl-1,2-oxazol-4-yl)-3-[(trimethyl-1H-pyrazol-1-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-6-methylpyridazine
2-[(4-fluorophenyl)methyl]-4-(1-methylcyclohexanecarbonyl)morpholine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)benzamide
1-[(2-{[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methyl]pyrrolidin-2-one
1-benzyl-N,N-dimethyl-5-{methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(1-methylcyclopropanecarbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 4-[4-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]benzoate
(3aS,7aR)-5-methyl-2-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(1R,5S,8R)-3-{[5-(2-methylpropyl)thiophen-2-yl]methyl}-3-azabicyclo[3.2.1]octan-8-ol
1-{3-[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]phenyl}pyrrolidin-2-one
N-(2,2-dimethyloxan-4-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-amine
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-methylquinoline
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
(3S,4R)-1-[2-(cyclohexylcarbamoyl)ethyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
(2S)-1-acetyl-N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
ethyl 4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazine-1-carboxylate
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(2-oxopyrrolidin-1-yl)propanamide
2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]benzonitrile
5-[(2-fluoro-4-methoxyphenyl)methyl]-5-[3-(2-methyl-4-phenylpiperazin-1-yl)-3-oxopropyl]pyrrolidin-2-one
2-(pyridin-4-ylmethyl)-9-[(2S)-2-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4-diazepane-6-carboxylic acid
1-methyl-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]-6-oxo-1,6-dihydropyridine-3-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-{3-[(pyridin-3-yl)amino]propyl}benzamide
2-[3-(dimethylamino)propyl]-9-[(1R,2R)-2-phenylcyclopropanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one