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methyl 1-methyl-3-(3-phenylpropanamido)-5-[(thiophen-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 2-[1-benzyl-8-(2,3-dihydro-1H-inden-2-yl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
5-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]pyrrolidin-2-yl}-3-phenyl-1,2,4-oxadiazole
2-[(4-methoxyphenyl)methyl]-1-[1-(5-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
1-cyclohexyl-3-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-3-(2-fluorophenyl)pyrrolidine-2,5-dione
3-(1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)benzoic acid
(1S,5R)-6-(3-propyl-1H-pyrazole-4-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-methyl-4-{4-[(4-phenylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}piperidin-4-ol
N-(2-chloro-4-fluoro-5-methylphenyl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
3-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1-[2-methoxy-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
1-{2-[(4-methyl-1,4-diazepan-1-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
1-cyclopentyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)-6-oxopiperidine-3-carboxamide
N-(2,3-dihydro-1H-inden-4-yl)-5-[({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amino)methyl]-1,3-thiazol-2-amine
N-[(2S,4R,6S)-2-ethyl-6-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]oxan-4-yl]benzamide
2-(2-phenoxyethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(methoxycarbonyl)benzoyl]piperidine-3-carboxylate
1-(2-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-2-oxoethyl)-1,4-dihydroquinolin-4-one
{1-[1-(2-phenylethyl)piperidin-3-yl]piperidin-4-yl}methanol
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrrolidin-2-one
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-methyl-6-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-(2-methoxyphenyl)-4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
4-(4-{[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenyl)but-3-yn-1-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-4,4,4-trifluoro-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}butanamide
1-(cyclopropylmethyl)-5-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-(thiophen-2-ylmethyl)propanamide
1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(3-methoxybenzoyl)piperazine
1-cyclopentyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-6-oxopiperidine-3-carboxamide
3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]propanamide
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-(1H-1,2,3,4-tetrazol-1-yl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-propoxypropanamide
(2R,4S)-4-hydroxy-1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidine-2-carboxylic acid
1-(2,3-dihydro-1H-inden-2-yl)-N-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-N-methylpiperidin-3-amine
methyl (2S,3S)-2-{[5-(tert-butylcarbamoyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridin-3-yl]formamido}-3-methylpentanoate
8-[(5-hydroxy-2-methoxyphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
(benzylsulfamoyl)[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]amine
{1-[(3-methylquinoxalin-2-yl)methyl]-4-(2-phenylethyl)piperidin-4-yl}methanol
3-chloro-2-[2-(1H-imidazol-1-yl)ethyl]-5-(trifluoromethyl)pyridine
N-[(1r,4r)-4-hydroxycyclohexyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxo-N-phenylacetamide
N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
4-(3-fluorophenyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzamide
2-[({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)amino]pyridine-4-carbonitrile
3-(2-ethyl-3-methyl-1-benzofuran-7-yl)-1-(3-hydroxypropyl)-1-(pyridin-3-ylmethyl)urea
1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-8-(4,4,4-trifluorobutan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(5-ethylfuran-2-yl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide