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3-(2-{2-[(4-fluorophenyl)methyl]morpholin-4-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(piperazine-1-carbonyl)benzene-1-sulfonamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N,5-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
1-(4-methoxybenzoyl)-4-(3,3,4,4,4-pentafluorobutyl)piperazine
cyclopentyl 4-({[3-(1H-1,2,4-triazol-1-yl)propyl]carbamoyl}amino)benzoate
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
N-[2-(2-fluorophenyl)-1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}ethyl]-N-methylthiophene-3-carboxamide
1-cyclohexyl-4-(2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazin-2-one
3-{[(1-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
[(3-{[1-(ethanesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-3-ylmethyl)amine
N-cyclohexyl-3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-[4-(butan-2-yloxy)-3-chloro-5-methoxyphenyl]-1H-imidazole
N-[(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]propanamide
1-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}ethan-1-one
1-ethyl-4-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]pyrrolidin-2-one
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-4-methoxybenzene-1-sulfonamide
N-(cyclopropylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-propylpiperidine-3-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}pyrrolidine-2-carboxamide
5-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1-(furan-3-ylmethyl)-4-phenyl-1H-imidazole
(1R,5S)-3-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octane
2-[8-(1,3-benzothiazol-2-ylmethyl)-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N-{[7-(2-cyclohexylacetyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
(2S)-2-[(3-methyl-5-propyl-1-benzofuran-2-yl)formamido]propanamide
3-(furan-2-yl)-1-{3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}propan-1-one
{3-[2-(1-phenylethyl)-1H-imidazol-1-yl]phenyl}methanol
(2S)-2-amino-1-[3-(3-chlorophenoxy)azetidin-1-yl]-3-hydroxypropan-1-one
1-[2-(dimethylamino)ethyl]-5-(3-methylfuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-butyl-2-{N-methyl-1-[4-(4H-1,2,4-triazol-4-yl)phenyl]formamido}acetamide
3-{2-oxo-2-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}imidazolidine-2,4-dione
1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
4-[5-(2-fluorobenzoyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
N-(furan-2-ylmethyl)-4-[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
2-({[3-fluoro-4-(trifluoromethyl)phenyl]carbamoyl}amino)hexanamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-6,7-dimethoxy-N,4-dimethylquinolin-2-amine
3-[3-(piperidine-1-carbonyl)-1-[3-(pyridin-3-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
ethyl 1-[1-(5-phenyl-1,2,4-triazin-3-yl)piperidin-4-yl]piperidine-4-carboxylate
2-[3-(2-fluorophenoxy)azetidine-1-carbonyl]benzene-1,3-diol
4-ethyl-3-(1-{[4-(trifluoromethyl)pyridin-3-yl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-ethyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyrimidine-5-carboxamide
5-(2-chlorophenoxymethyl)-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
4-benzyl-3-butyl-1-{2-[3-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{3-[7-(but-3-enoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]-1,2,4-oxadiazol-5-yl}benzonitrile
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-4-methyl-1,2,3-thiadiazole
7-chloro-4-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 5-({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
(4S,4aS,8aR)-1-(2-cyclopropyl-1,3-benzoxazole-6-carbonyl)-4-phenyl-decahydroquinolin-4-ol
dimethyl[3-({5-[6-(trifluoromethyl)pyridin-3-yl]pyridin-2-yl}oxy)propyl]amine
N-(cyclohexylmethyl)-1-[2-(dimethylamino)ethyl]-6-methyl-4-oxo-2-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
7-cyclopropanecarbonyl-N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine