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1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
2-(methylsulfanyl)-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyrimidine
N-(pyridin-2-ylmethyl)-1-(2-{2-[3-(trifluoromethyl)phenyl]acetamido}ethyl)-1H-1,2,3-triazole-4-carboxamide
(3aR,6aR)-2-cyclopentanecarbonyl-5-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-N'-[2-(propan-2-yl)phenyl]butanediamide
1-methyl-5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
4-[({dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)methyl]-1-methyl-1,2,3,4-tetrahydroquinolin-2-one
2-{4-[(3-methyl-1H-indol-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4-(2-phenylethyl)piperidin-4-yl]methanol
4-({[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}amino)-2-methoxypyridine-3-carbonitrile
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}propan-1-one
(2R,3S,6R)-3-phenyl-5-(2-phenylethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[8-(3-methoxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]-4,6-dimethylpyridine-3-carbonitrile
2-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-amine
[2,2-dimethyl-3-(morpholin-4-yl)propyl](furan-2-ylmethyl)(thiophen-3-ylmethyl)amine
3-[(4-ethylpiperazin-1-yl)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-[1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
2-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-1,2-dihydroisoquinolin-1-one
N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
1-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
N-[1-(methoxymethyl)cyclopentyl]-3-(pyridin-4-yl)propanamide
4-{4-[2-(3-chlorophenyl)acetyl]piperazin-1-yl}-2-[2-(4-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-2H-1,3-benzodioxole-5-carboxamide
4-[(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]piperidine
3-[3-(4-fluorophenyl)oxolan-3-yl]-5-(3-methyl-1H-pyrazol-5-yl)-1,2,4-oxadiazole
ethyl 4-[2-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-5-oxopyrrolidin-1-yl]piperidine-1-carboxylate
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidin-3-yl]acetamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
(2S,4S)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N,N-diethyl-4-(1-methylcyclopropaneamido)pyrrolidine-2-carboxamide
N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-1H-1,2,3-benzotriazole-5-carboxamide
2-[methyl(pyridin-2-ylmethyl)amino]-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
2-methyl-N-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[4-(1H-imidazol-1-yl)benzoyl]pyrrolidine-2-carboxamide
4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]benzamide
2,2-dimethylpropyl 4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
N-[(1S,2S)-2-hydroxycyclohexyl]-3,5-dimethyladamantane-1-carboxamide
3-[(2-fluorophenyl)formamido]-N-[(4-phenyloxan-4-yl)methyl]propanamide
1-[(2-ethylpyrimidin-5-yl)methyl]-N,N-dimethylpiperidin-3-amine
8-[(3-methoxyphenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-cyclopentyl-8-(5-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2-(trifluoromethyl)benzamide
3-({4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
2-methoxy-3-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pyrazine
3-(2,5-dioxoimidazolidin-4-yl)-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]propanamide
N-benzyl-1-[1-(5-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
9-ethyl-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
N-[3-(3-ethylphenoxy)propyl]-N-methylquinoxaline-5-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)(methyl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine