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N,N-diethyl-1-{1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}pyrrolidin-3-amine
4-benzyl-1-(naphthalen-1-ylmethyl)-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-chlorophenyl)-4-[2-(propan-2-yl)pyrimidine-4-carbonyl]piperazin-2-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(pyrrolidin-1-yl)propan-1-one
7-(cyclobutylsulfamoyl)-N-(propan-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
5,6-dimethyl-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]thieno[2,3-d]pyrimidine
2-(3,4-dichlorophenyl)-4-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]morpholine
6-{4-[(2-methoxypyridin-3-yl)methyl]piperazin-1-yl}pyrazine-2-carboxamide
5-amino-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1H-pyrazole-3-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidine
4-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)-N-(2-phenylethyl)piperidine-1-carboxamide
2-ethyl-N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}pyrimidine-5-carboxamide
5-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazol-3-ol
N-[2-(dimethylamino)ethyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-[4-(dimethylamino)phenyl]-1-[3-(2-methoxyphenoxy)azetidin-1-yl]ethan-1-one
6-phenyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-phenyl-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1,2-oxazole-3-carboxamide
1-[2-(4-methoxyphenyl)ethyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
N-ethyl-1-(furan-2-ylmethyl)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-4-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(1H-imidazol-1-yl)propyl]-2,7,8-trimethylquinoline-4-carboxamide
N-({1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-4-yl}methyl)acetamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}quinoxaline-5-carboxamide
4-({2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-benzyl-9-[2-(morpholin-3-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-{4-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
3-(4-methyl-1H-pyrazol-5-yl)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidine
4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N,N-dimethylbenzene-1-sulfonamide
2-(5-acetylthiophen-3-yl)-N-{2-[(2-chlorophenyl)formamido]ethyl}acetamide
2-[1-(3-methylbutyl)-2,4-dioxo-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
2-(2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-benzotriazole
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]but-3-en-1-one
2-{4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-1-yl}pyrazine
2-[methyl(2-phenylethyl)amino]-N-[2-(pyrrolidin-1-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(3-fluorophenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
N-(2-methoxyethyl)-N-methyl-3-[(oxan-3-ylmethyl)sulfamoyl]benzamide
3-(3-methylphenoxy)-1-[3-(methylsulfanyl)propyl]azetidine
5-ethyl-5-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-[2-(4-methoxyphenyl)ethyl]imidazolidine-2,4-dione
2-{[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}quinolin-8-ol
6-(2-aminoethyl)-N,2-dimethyl-N-[(1R)-1-(naphthalen-1-yl)ethyl]pyrimidin-4-amine
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-4-methoxypyrimidine
4-(5-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
2-(4-{[3-(furan-2-yl)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
6-({4-[2-(5-methylfuran-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)pyrimidin-4-ol
4-methoxy-6-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]pyrimidin-2-amine