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5-methyl-N-[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(2-{1-[4-(2-oxopiperidin-1-yl)butanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
[(2S,4R)-4-(dimethylamino)-1-({2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}methyl)pyrrolidin-2-yl]methanol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
3-(2,5-dimethoxyphenyl)-1-{5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidine
(1S,5R)-6-(cyclobutylmethyl)-3-[(2,3-difluoro-4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(4aS,8aR)-1-(2-aminoethyl)-6-{[2-(2-hydroxyethoxy)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
2-{5-[1-(ethylsulfanyl)ethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}pyridine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-(1H-pyrazol-4-yl)butan-1-one
1-[(4R)-3-methyl-1,3-thiazolidine-4-carbonyl]-4-[(2-methylphenyl)sulfanyl]piperidine
5-{[2-(morpholin-4-yl)ethyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
3-methyl-5-{2-oxo-2-[2-(trifluoromethyl)morpholin-4-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3R,5S)-1-benzyl-5-(3-fluorophenoxymethyl)-N-[2-(1H-imidazol-4-yl)ethyl]piperidine-3-carboxamide
8-(piperidin-4-yl)-3-{3-[4-(propan-2-yl)piperazin-1-yl]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-ethyl-2-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]propane-1,3-diol
3,4,7-trimethyl-N-[(3R,4R)-4-(4-methylpiperazin-1-yl)oxolan-3-yl]-1H-indole-2-carboxamide
2-[3-methyl-4-(morpholin-4-yl)benzoyl]-2,7-diazaspiro[4.5]decane
(1R,7S)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine
4-{imidazo[1,2-a]pyridine-3-carbonyl}-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
2-({[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}(pyridin-3-ylmethyl)amino)butan-1-ol
2-(4-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenoxy)ethan-1-ol
3-{2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
N-{3-[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]-4-methoxyphenyl}acetamide
3-benzyl-1-[3-(hydroxymethyl)quinolin-2-yl]piperidine-3-carboxylic acid
(4aS,7aR)-1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-4-cyclopropyl-1-{[5-(methylcarbamoyl)furan-2-yl]methyl}pyrrolidine-3-carboxylic acid
4-{2-[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethyl}morpholine
N-cyclobutyl-4-{[(2S)-pyrrolidin-2-ylmethyl]sulfamoyl}benzamide
N-[2-(dimethylamino)ethyl]-4-(pyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
5-(2,4-difluorophenoxymethyl)-N-(oxan-4-ylmethyl)-1H-pyrazole-3-carboxamide
2-{3-oxo-9-[(2,3,4-trifluorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
(1S,5R)-3-(1H-indol-5-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[2-(2-methoxyphenyl)acetyl]-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
3-(2-oxopyrrolidin-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
N-{[3-(4-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-(2-methyl-1H-imidazol-1-yl)propanamide
(1S,5R)-6-(dimethyl-1,2-oxazole-4-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
6-({4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-3-carbonyl]piperidin-4-yl}oxy)quinoline
N-(cyclohex-1-en-1-ylmethyl)-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-methyl-1H-indol-1-yl)propanamide
6-{4-[(dimethylamino)methyl]phenyl}-N-(propan-2-yl)pyridazin-3-amine
4-(4-methylpiperazin-1-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)pentanamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
7-(2-phenylethyl)-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-3-methylthiophene-2-carboxamide
N'-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N,N-dimethyl-N'-(oxolan-2-ylmethyl)butanediamide
2-(4-{[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]methyl}phenyl)ethan-1-amine
5-chloro-2-methoxy-4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridine
3-{5-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
6-[4-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyrimidin-4-amine