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4-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1λ6-thiane-1,1-dione
{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)(1,2-oxazol-3-ylmethyl)amine
4-benzyl-3-ethyl-1-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-1,4-diazepan-5-one
(1R,5R)-6-(1-hydroxynaphthalene-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
5-(3-methoxyphenyl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1,2,4-triazin-3-amine
N,8-dimethyl-N-(propan-2-yl)-2-[2-(pyridin-3-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-methyl-5-[(quinolin-8-yloxy)methyl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-oxopiperidin-1-yl)propanamide
4-chloro-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-2-propanamidobenzamide
methyl(1,2-oxazol-3-ylmethyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
{4-[3-(oxan-4-yl)-1-propyl-1H-1,2,4-triazol-5-yl]phenyl}methanamine
(4aS,7aR)-1-(4-ethylbenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(4aS,8aR)-6-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-decahydro-1,6-naphthyridin-4a-yl]methanol
methyl 2-[(1-ethyl-1H-pyrazol-3-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
4-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]imidazolidin-2-one
(4aR,8aS)-1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridine
6-(benzyloxy)-1-cyclohexyl-4-(6-methylpyridine-2-carbonyl)-1,4-diazepan-2-one
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-4-(4H-1,2,4-triazol-4-yl)benzamide
3-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
4-({methyl[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)-1H-pyrazole-3-carboxylic acid
4-[(1-methoxybutan-2-yl)amino]-5-methyl-N-[2-(methylsulfanyl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-cyclopropyl-N-{1-[1-(1-methylpiperidine-3-carbonyl)piperidin-4-yl]-2-phenylethyl}pyridine-2-carboxamide
7-[3-(1H-pyrazol-4-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
{4-[2-(methylamino)-4-(4-methylphenyl)pyrimidin-5-yl]phenyl}methanol
N-cyclohexyl-1-cyclopropyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
11-[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
4-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-1,2,3,4-tetrahydroquinolin-2-one
7-[2-(2-methyl-1H-indol-3-yl)acetyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-({2-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2-acetamido-3-methylbutanamide
1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
1-methyl-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
3-[(1-ethyl-1H-pyrazol-3-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-hydroxy-1-(2-phenylethyl)-3-{[4-(propan-2-yl)piperazin-1-yl]methyl}piperidin-2-one
1-(4-methoxyphenyl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-2-one
9-[2-(3-hydroxyphenyl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({[(3R,4R)-4-(hydroxymethyl)-1-[6-(morpholin-4-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[2-(cyclohexylsulfanyl)ethyl]-3-[1-(propan-2-yl)-1H-pyrazol-5-yl]urea
5-{5-[5-(methoxymethyl)thiophen-2-yl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-3-(dimethyl-1,2-oxazol-4-yl)-N-methylpropanamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}acetamide
4-{4-[(4-methoxy-2,5-dimethylphenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
2-{[4-(2-chloro-4-fluorophenyl)phenyl]methoxy}ethan-1-amine
3-(pyrrolidine-1-carbonyl)-2-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]pyridine
N-cyclopropyl-8-fluoro-N-(1,3-thiazol-5-ylmethyl)quinoline-2-carboxamide
5-[2-({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3,4-thiadiazol-2-amine
3-[1-(5-aminopyrazin-2-yl)-1H-1,3-benzodiazol-2-yl]propan-1-ol
N-[(2-phenoxypyridin-3-yl)methyl]-2-(pyridin-4-yl)acetamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(pyrrolidin-3-yl)benzamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-ethyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide