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N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]-1,3-thiazole-5-carboxamide
1-[(2-fluorophenyl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-[2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-oxoethyl]-1,2-dihydrophthalazin-1-one
2-(hydroxymethyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,3-benzodiazole-5-carboxamide
N-(4-{[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenyl)acetamide
N-(3-acetylphenyl)-3-(morpholin-4-yl)piperidine-1-carboxamide
2-(4-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
2-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-(quinoxalin-6-ylmethyl)benzamide
2-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl](thiophen-3-ylmethyl)amino}butan-1-ol
2-[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]-2-(2,3-dihydro-1,4-benzodioxin-6-yl)acetic acid
7-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}-1,2,3,4-tetrahydroquinoxalin-2-one
(3R,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
ethyl 1-[5-(methoxymethyl)thiophene-2-carbonyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
1-ethyl-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
8-fluoro-2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,4-dihydroquinolin-4-one
N-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-yl}pyrimidin-2-amine
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-(2-phenylethyl)piperidin-2-one
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)pyrrolidine-1-sulfonamide
N-(furan-3-ylmethyl)-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-ethyl-8-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[1-(pyridin-2-yl)propan-2-yl]propanamide
2-[methyl(2-phenylethyl)amino]-N-[2-(pyridin-2-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-[(8-chloronaphthalen-1-yl)sulfonyl]-2-(trifluoromethyl)morpholine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
methyl 6-{[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]carbamoyl}pyridine-3-carboxylate
2-chloro-6-fluoro-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}benzamide
N-[3-(3-methylphenyl)phenyl]-1-(oxane-4-carbonyl)piperidine-3-carboxamide
2-methoxy-N-[(2-methoxyphenyl)methyl]-N-propylbutanamide
N-[(2R,3R)-2-hydroxy-1'-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
5-(2-methoxypyridine-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
7-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
5-[(4-methyl-3-phenylpiperazin-1-yl)methyl]quinoline
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(propan-2-yl)acetamide
3-[4-(1H-pyrazol-5-yl)benzoyl]-3,9-diazaspiro[5.5]undecane
(3aR,6aR)-N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(2S,4S)-4-(4-{2-[(3-chlorophenyl)formamido]propan-2-yl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
2-ethyl-9-{2-methyl-3-oxo-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
2-{[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole
N-cyclopropyl-1-{1-[4-(4-fluorophenyl)-4-oxobutanoyl]piperidin-4-yl}piperidine-4-carboxamide
6-methyl-1-(3-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
(1S,3R)-3-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]cyclohexan-1-amine
1-(2-methoxyphenyl)-4-[(2S)-2-(methylamino)propanoyl]piperazin-2-one
2-[4-(4-{[(5-amino-1H-1,2,4-triazol-3-yl)methyl]amino}piperidin-1-yl)-6-methylpyrimidin-2-yl]phenol
N-[4-(4-{[2-methyl-2-(morpholin-4-yl)propyl]amino}piperidin-1-yl)phenyl]-3-phenylpropanamide
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
methyl (1R,3S,3aR,6aS)-3-(1,5-dimethyl-1H-pyrazol-4-yl)-1-(2-methoxy-2-oxoethyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-[(2,4-dimethylphenyl)methyl]-4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidine