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1-(4-fluorophenyl)-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]cyclopropane-1-carboxamide
N-(2-ethoxyethyl)-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}acetamide
1-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-4-(2-methylpropyl)-1,4-diazepan-5-one
2-(4-{[benzyl(methyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N,N-bis(2-hydroxyethyl)acetamide
3-[1-(cyclohexylmethyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
3-(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-1-ol
N-({8-[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
methyl 2-{[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]amino}acetate
N-({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)-N-(pyridin-2-ylmethyl)cyclopropanamine
3-ethyl-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-ol
4-(1-{2-[methyl(pyridin-3-ylmethyl)amino]acetyl}piperidin-3-yl)benzoic acid
N-(2-methylpropyl)-1-[(1s,4s)-4-{[(2,4,5-trimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
N-[2-(pyridin-2-ylsulfanyl)ethyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
5-{5-[1-(4-chlorophenyl)cyclopropyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N'-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N'-(oxolan-2-ylmethyl)butanediamide
(5-{[ethyl({[2-(prop-2-en-1-yloxy)phenyl]methyl})amino]methyl}furan-2-yl)methanol
3-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
ethyl 3-benzyl-1-(3-methylbut-2-enoyl)piperidine-3-carboxylate
2-methyl-N-(1,3-thiazol-2-yl)-3-[3-(1H-1,2,4-triazol-1-yl)propanamido]benzamide
(4aR,8aR)-2-{imidazo[1,2-a]pyrimidine-2-carbonyl}-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
6-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-3-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}propanamide
(3R,4R)-4-cyclobutyl-3-methyl-1-(4,4,4-trifluorobutyl)piperidin-4-ol
N-methyl-3-(2-oxo-1,2-dihydropyridin-1-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
(2S,4R)-4-amino-N-methyl-1-[3-(4-methylbenzenesulfonyl)propanoyl]pyrrolidine-2-carboxamide
3-(1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
(1S,3R)-3-amino-N-(2,3-dihydro-1H-inden-4-yl)cyclopentane-1-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(quinolin-4-ylmethyl)piperidin-3-yl]propanamide
3-{2-[4-(4-acetylphenyl)piperazin-1-yl]-2-oxoethyl}-3-(2-chlorophenyl)-1-methylpyrrolidine-2,5-dione
2-(4-ethoxyphenyl)-1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
2-ethyl-9-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(4-ethylpiperazin-1-yl)-1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]ethan-1-one
(3S)-3-ethyl-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)morpholine
4-[4-(4-methoxy-4-phenylpiperidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
1-[1-(5-chloro-2-methylpyrimidine-4-carbonyl)piperidin-4-yl]piperidin-4-ol
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
(2S,4S)-4-amino-1-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-2-carboxylic acid
N-(5-acetyl-2-ethoxyphenyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
2-(pyridin-4-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidine-5-carboxamide
3-{2-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-oxoethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-6-(pyrrolidin-1-yl)pyrimidin-2-amine
4-(2,5-dimethylbenzoyl)-1-(4-methoxyphenyl)-5-methylpiperazin-2-one
3-{[5-(4,5-dimethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-(propan-2-yl)-1,2,4-oxadiazole
{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine