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2-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
dimethyl(3-{2-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-4-methoxy-N-methylbenzamide
1-methyl-3-phenyl-5-(thiophen-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
1-(2-methyloxolane-2-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
[(3R,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-N-[(4-methyl-1,3-thiazol-2-yl)methyl]pyrimidin-2-amine
N-(2-methoxyethyl)-5-(methoxymethyl)-N-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(pyrrolidin-3-yl)-N-[3-(trifluoromethoxy)phenyl]benzamide
8-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[(2S,4R,6R)-2-(3-chloro-5-fluoro-4-methoxyphenyl)-6-(propan-2-yl)oxan-4-yl]acetamide
1-cyclobutanecarbonyl-N-[(5-methoxy-1H-indol-2-yl)methyl]piperidine-4-carboxamide
1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
methyl 4-[2-(3-methoxypropyl)piperidine-1-carbonyl]benzoate
4-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzene-1-sulfonamide
4-(4-phenoxybutyl)-1,4-oxazepan-5-one
1-[2-(3-fluorophenyl)ethyl]-N-methyl-N-[2-(oxan-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-methoxypyridine
N-[(1-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl)methyl]acetamide
2-(1-benzofuran-2-yl)-2-(morpholin-4-yl)acetic acid
2-(2-{4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}ethoxy)ethan-1-ol
1-({2-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)piperidin-4-ol
1-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-{5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamido]-2-methylphenyl}-3-methylbenzamide
(cyclopropylmethyl)({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
5-(3-{3-[(2-fluorophenyl)methoxy]azetidin-1-yl}-3-oxopropyl)imidazolidine-2,4-dione
9-[(2S)-2-amino-4-(methylsulfanyl)butanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-chloro-1,3-dimethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1H-pyrazole-5-carboxamide
N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}oxolane-3-carboxamide
8-chloro-2-{[4-(1,3-thiazol-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
4-{[(4-fluorophenyl)methyl]sulfamoyl}-N-(2-hydroxypropyl)benzamide
3-[(2-methylphenyl)methyl]-1-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperidine-3-carboxylic acid
N-{[7-methoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)oxolane-2-carboxamide
5-cyclopropyl-N-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,3-oxazole-4-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[5-(methoxymethyl)furan-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-(2,3-dihydro-1H-inden-2-yl)-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(furan-2-ylmethyl)(2-hydroxyethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(2-methylbutan-2-yl)acetamide
8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(1H-indol-3-yl)ethyl]-5-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
1-(2-{4-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
{5-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-(adamantan-1-ylmethyl)-1-[(4-fluorophenyl)methyl]-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1-(morpholin-4-yl)ethan-1-one
(2S,4R)-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-N-methyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
N-[(3R,4S)-1-benzyl-4-propylpyrrolidin-3-yl]-3-methanesulfonylpropanamide
N-{1-[1-(3-hydroxy-2,2-dimethylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide