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4-(azepane-1-carbonyl)-2-(1-ethyl-1H-pyrazol-4-yl)-6-methylquinoline
N-[(4-fluorophenyl)methyl]-5-[(2-hydroxyethyl)(methyl)amino]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(5-chlorothiophen-2-yl)methyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
N-(2,2-difluoroethyl)-4-[(2-hydroxy-3-methoxypropyl)sulfamoyl]benzamide
5-(2-fluorophenoxymethyl)-N-[(1-hydroxycyclohexyl)methyl]-1H-pyrazole-3-carboxamide
7-(cyclopropylmethyl)-N,N-dimethyl-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[2-(pyridin-3-yloxy)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[1-(2-methoxyethyl)-7-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-1,3-benzodiazol-5-yl]cyclohexanecarboxamide
(1R,7S)-3-(2-ethylbutyl)-6-(4-methyl-1,4-diazepane-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-[2-(5-methylfuran-2-yl)ethyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
4-(3,5-difluoropyridine-2-carbonyl)-1-(4-methoxyphenyl)-3-methylpiperazin-2-one
8-(4-methyl-1H-imidazole-2-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
8-[(1-ethyl-1H-indol-4-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(2,3-dimethoxyphenyl)methyl]-N-methylthian-4-amine
2-cyclopentyl-9-[(2-methylpyrimidin-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-methoxy-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-4H-pyran-4-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-{5-[(2-methyl-1H-imidazol-1-yl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
3-methyl-4-(3-methyl-1H-pyrazole-5-carbonyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
4-(piperidin-1-yl)-N-[1-(1,3-thiazol-2-yl)propyl]butanamide
1-{2-[methyl({[3-(trifluoromethyl)phenyl]methyl})amino]ethyl}piperidin-2-one
4-{[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
8-[4-(dimethylamino)pyrimidin-2-yl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-yl)acetamide
7-methyl-2-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
9-(2-methoxypyridine-4-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide
8-[1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carbonyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-[5-(ethanesulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1-(4-hydroxypiperidin-1-yl)propan-1-one
2-cyclopropyl-8-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-ethoxypropan-1-one
2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-4,5,6,7-tetrahydro-1,3-benzothiazole
N-(3-chloro-4-fluorophenyl)-N'-(furan-2-ylmethyl)-N'-(pyridin-4-ylmethyl)propanediamide
5-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-4-methylpyrimidine
1-{2-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-(4-hydroxy-3-methoxyphenyl)-1,3,8-triazatricyclo[7.4.0.02,7]trideca-2(7),8-dien-4-one
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-N-phenylpyrimidin-2-amine
N-{[7-(5-ethylpyrimidin-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
5-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridine-3-carboxamide
2-{2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(2-{[4-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)piperazin-1-yl]methyl}phenyl)methanol
3-{methyl[1-(pyridin-3-yl)propyl]carbamoyl}benzoic acid
5-({2-[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole
2-acetyl-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)benzamide
ethyl 1-{[3-(ethoxycarbonyl)-1H-pyrazol-4-yl]methyl}-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
2-(2,4-difluorophenoxy)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
4-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-4-oxobutane-1-sulfonamide
4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-2-(4-methylpentyl)morpholine