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2-[2-({methyl[2-(2-oxopiperidin-1-yl)ethyl]amino}methyl)phenoxy]acetic acid
2-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}quinolin-8-ol
3-benzyl-8-[(3-hydroxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-1-(2-fluorophenyl)cyclopropane-1-carboxamide
N-[2-(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{1-[5-(3-fluoro-5-methylphenyl)-4-phenyl-1H-imidazol-1-yl]ethyl}-4-methyl-4H-1,2,4-triazole
[5-({[2-(dimethylamino)ethyl][(2-methylphenyl)methyl]amino}methyl)furan-2-yl]methanol
6-(2-fluorophenyl)-N-[2-(6-hydroxypyrimidin-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-2-[3-(2-fluorophenyl)-4-methyl-1H-pyrazol-1-yl]acetamide
1-(2-methoxy-5-{[methyl(oxan-4-yl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
N-{[3-methyl-7-(thiophene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-2-oxopentanamide
N-[2-(dimethylsulfamoyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-2-methoxybenzamide
N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
methyl 3-{3-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]piperidine-1-carbonyl}benzoate
(3S,4R)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-(morpholine-4-carbonyl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyridin-4-amine
5-(2-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
(3S,5R)-N3-cyclohexyl-N5-(2,3-dihydro-1H-inden-5-yl)piperidine-3,5-dicarboxamide
1-benzyl-3-(2-methoxyethyl)-8-[3-(5-methylfuran-2-yl)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (2S)-1-(2-{1-[2-(1H-imidazol-1-yl)ethyl]-2,5-dioxo-3-phenylpyrrolidin-3-yl}acetyl)pyrrolidine-2-carboxylate
3-{imidazo[1,2-a]pyridin-2-yl}-1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]propan-1-one
2-amino-N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-ethyl-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
[3-(1H-indol-1-yl)propyl](4,4,4-trifluorobutan-2-yl)amine
methyl 6-[8-(3-hydroxypropyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxylate
4-[(2S)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidine-2-carbonyl]morpholine
N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
9-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-[2-(1-benzyl-1H-1,2,4-triazol-5-yl)phenyl]-1λ6-thiomorpholine-1,1-dione
5,6-dimethoxy-2-(3-methoxypropyl)-1,2-dihydroisoquinolin-1-one
5-chloro-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-methyl-N-(pyridin-3-ylmethyl)-1,3-thiazole-4-carboxamide
N-[(2-fluorophenyl)methyl]-1-methyl-5-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(thiophen-2-yl)-1-[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]ethan-1-one
5-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]quinoxaline
1-methyl-5-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(2-phenoxyethyl)-2,8-diazaspiro[4.5]decan-3-one
2-(3-methyl-3-phenylpiperidin-1-yl)-1,3-thiazole-4-carboxamide
N-[2-(2-chlorophenyl)ethyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(4-{pyrazolo[1,5-a]pyridin-7-yl}phenoxy)ethanimidamide
4-[4-(3-cyclohexylpropanoyl)piperazin-1-yl]-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-(furan-2-ylmethyl)-5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N,N-dimethyl-2-[({thieno[2,3-d]pyrimidin-4-yl}amino)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(1R,5S)-3-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]-3,8-diazabicyclo[3.2.1]octane
6-(4-methyl-1H-pyrazol-1-yl)-2H-1,3-benzodioxole-5-carboxamide
1-[4-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazin-1-yl]ethan-1-one
3-(3-fluorophenoxymethyl)-1-[2-(1H-imidazol-5-yl)ethyl]-5-(oxan-2-yl)-1H-1,2,4-triazole
11-methyl-5-[2-(1-methylpiperidin-2-yl)ethyl]-8-thia-3,5,10-triazatricyclo[7.4.0.02,7]trideca-1(13),2(7),3,9,11-pentaen-6-one
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl){[5-(pyridin-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
6-ethyl-5-methyl-N4-[3-(4-methyl-1H-pyrazol-1-yl)propyl]pyrimidine-2,4-diamine