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1-[1'-(2-hydroxy-5-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-(4-aminobutyl)-5-(2-chlorophenyl)-2-methylfuran-3-carboxamide
4-{4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]piperidin-1-yl}-N-[2-(morpholin-4-yl)ethyl]benzamide
N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
N-methyl-N-(propan-2-yl)-2-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-ethyl-2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)pyrimidin-4-amine
2-methylpropyl N-[(3R,5S)-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)pyrrolidin-3-yl]carbamate
N3-methyl-1-(2-methylpropyl)-4-oxo-N3-(2-phenylethyl)-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-{[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrazole
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2-(trifluoromethyl)-1H-1,3-benzodiazole-5-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)propanamide
1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-3-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}urea
1-(3-{[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]methyl}phenyl)ethan-1-one
4-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]quinoline
1-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-phenylpiperidin-4-yl}ethan-1-one
4-hydroxy-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-[(phenylsulfanyl)methyl]pyrimidine-5-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-1-methylazepane-2-carboxamide
(3S)-3-({2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)azepan-2-one
1-(carbamoylmethyl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]piperidine-3-carboxamide
2,3-dimethyl-6-(1-methylazepane-2-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
2-(pyridin-3-yl)-4-[(3,4,5-trimethoxyphenyl)methyl]morpholine
propyl 2-{4-[benzyl(methyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}acetate
1-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]urea
6-{4-[1-(morpholin-4-yl)ethyl]phenyl}pyridin-2-amine
5-(4-fluorophenyl)-N-[2-(pyridin-3-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(3-chloro-4-methylphenyl)-2-(acetamidomethyl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
1-[cyclohexyl(methyl)amino]-3-(2-{[(3-ethoxypropyl)amino]methyl}phenoxy)propan-2-ol
1-[3-(piperidin-3-yl)benzoyl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
4-(3-{2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl}propoxy)benzamide
3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-ol
3-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-5-methyl-1H-indole
2-phenyl-1-({3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}methyl)-1H-imidazole
4-ethyl-1-methyl-3-({1-[(7-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-chloro-1-methyl-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-1H-indole-2-carboxamide
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(cyclopropylsulfamoyl)-5-(isoquinolin-5-yl)benzoic acid
8-(cyclohex-3-en-1-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[5-carbamoyl-2-(2-methylpiperidin-1-yl)phenyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-(methoxymethyl)-5-{[3-(4-methoxyphenoxymethyl)piperidin-1-yl]methyl}pyrimidine
2-(2-methylphenyl)-1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidine
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
3-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}oxy)-N-(2-phenylethyl)benzamide
3-(1-benzyl-1H-imidazol-2-yl)-1-(1H-pyrrole-2-carbonyl)piperidine
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-methyl-N-(propan-2-yl)acetamide
4-[4-(furan-2-ylmethyl)piperazine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
3-methyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
methyl 1-ethoxy-8-[3-(1H-indol-3-yl)propanoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-benzyl-N-methyl-3-{1-[2-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}propanamide
N-(1-benzylpiperidin-4-yl)-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine