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4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine
3-(4-cyclopentyl-1,4-diazepane-1-carbonyl)-4-fluorobenzene-1-sulfonamide
2-(1-{[3-(cyclopentyloxy)phenyl]methyl}pyrrolidin-2-yl)ethan-1-ol
N,7,8-trimethyl-N-(propan-2-yl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-methylpiperidin-2-one
8-(2-ethoxypyridine-3-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3-methoxyphenyl)methyl]-N-methyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2,5-dimethoxyphenyl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
2-(adamantan-1-yl)-4-hydroxy-N-[2-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
6-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-benzyl-4-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-7-propyl-2,7-diazaspiro[4.5]decan-6-one
6-cyclopropyl-N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]pyrimidin-4-amine
1-[(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carboxamide
5-[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]quinoxaline
1-(1-benzothiophene-2-carbonyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
2-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl)methyl]cyclobutanecarboxamide
6-{[(1R,3R)-3-aminocyclopentyl]amino}-5-chloropyridine-3-carboxylic acid
N-(3,5-dimethoxyphenyl)-3-[1-(furan-3-carbonyl)piperidin-3-yl]propanamide
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-1-phenyl-1H-1,2,3-triazole-4-carboxamide
3-({1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-4-yl}methyl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl})amine
(3S,4S)-4-{[2-(3-ethylphenoxy)ethyl](methyl)amino}-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-ol
methyl 2-{[2-(methoxymethyl)-1-methyl-5-(2-phenylacetamido)-1H-1,3-benzodiazol-7-yl]formamido}-4-(methylsulfanyl)butanoate
(2S,4R)-4-amino-N,N-diethyl-1-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]pyrrolidine-2-carboxamide
1-(but-2-ynoyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
4-{5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-2-amine
(2R)-2-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-one
N-(4-methoxyphenyl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-3-amine
(1R,2R,6S,7S)-4-(3-ethyl-1H-indole-2-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
3-(3-hydroxy-3-methylbutyl)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]benzamide
2-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(2-hydroxy-3-methoxypropyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
2-methoxy-4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-cycloheptyl-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-amine
4-[3-(ethanesulfonyl)phenyl]-1H-imidazole
1-(1-benzylpiperidin-4-yl)-N-(3-hydroxypropyl)piperidine-3-carboxamide
2-(5-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
N-[(3S)-1-(5-methanesulfonyl-2-methylpyrimidin-4-yl)pyrrolidin-3-yl]acetamide
3-[4-(3-methylphenyl)piperazin-1-yl]-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]propan-1-one
(3R,5S)-1-[(4-hydroxyphenyl)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
N-[2-hydroxy-2-(pyridin-4-yl)ethyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
9-[(4-acetylphenyl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3aR,5S,6S,7aS)-2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-octahydro-1H-isoindole-5,6-diol
(1R,5R)-3-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane