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8-(butan-2-yl)-3-ethyl-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-dimethyl-2-{[(7-methyl-1-benzofuran-2-yl)formamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)(pentan-3-yl)amine
4-(3-fluoro-4-methylbenzenesulfonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[2-(propan-2-yl)pyrimidine-4-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(4aS,8aR)-6-(dimethyl-1,3-oxazole-5-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-[(3,5-dimethylphenyl)methyl]-4-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperazin-2-one
2-{1-methyl-5-[4-(propan-2-yl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
8-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(2,4-diethoxy-3-methylphenyl)methyl]azepan-4-amine
N-[3-(1H-imidazol-1-yl)propyl]-2-(methoxymethyl)-6-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
1-(3-fluorophenyl)-6,6-dimethyl-N-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
(1S,5R)-3-[(1-ethyl-1H-imidazol-2-yl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
N-[4-(pyridin-2-yl)butyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[6-(pyridin-4-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-(4-chloro-2-fluorophenyl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-4-(3-cyclohexylpyrrolidine-1-carbonyl)-1,3-oxazole
N'-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-N,N-dimethylbutanediamide
5,6-dimethyl-2-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
(3R,4R)-1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
N,6-dimethyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
(1S,3R)-N1-(2,1,3-benzothiadiazol-5-ylmethyl)-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
2-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(furan-2-ylmethyl)amino]butan-1-ol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-[2-(dimethylamino)ethyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
(4aS,8aS)-2-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-5-ethyl-1,3-oxazole-4-carboxamide
(4-{[(4-methanesulfonylmorpholin-2-yl)methyl]amino}quinazolin-2-yl)methanol
2-{1-methyl-4-[(6-methylpyridin-2-yl)methyl]-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
2-(hydroxymethyl)-N-[(1R,2S)-2-phenylcyclohexyl]-1H-1,3-benzodiazole-5-carboxamide
2-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(1H-indol-1-ylmethyl)-N-[(5-methylpyrazin-2-yl)methyl]-1H-pyrazole-3-carboxamide
1-(2H-1,3-benzodioxol-5-yl)-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)piperidin-4-amine
2-{1-[(4-fluorophenyl)methyl]-4-(quinolin-8-ylmethyl)piperazin-2-yl}ethan-1-ol
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-methyl-5-({3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
5-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
5-[4-hydroxy-1-(2-methylpropyl)piperidin-4-yl]-N-(2-methoxyphenyl)-1-benzofuran-2-carboxamide
5-[4-(1H-pyrazol-1-yl)phenyl]pyridine-2-carbonitrile
2-{4-[2-(7-fluoro-2-methyl-1H-indol-3-yl)acetyl]piperazin-1-yl}pyridine-3-carbonitrile
(1-{1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methanamine
3-{[methyl({[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazol-4-yl]methyl})amino]methyl}phenol
2-(1,4-dioxan-2-ylmethyl)-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
5-(3-methoxypyrazin-2-yl)-8-methylquinoline
methyl N-{[({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)carbamoyl]methyl}carbamate
1-[2-(dimethylamino)ethyl]-N-{[5-(dimethylcarbamoyl)furan-2-yl]methyl}-5-oxopyrrolidine-3-carboxamide
3-{[2-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-3-(4H-1,2,4-triazol-4-yl)benzamide