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3-(1-butyl-1H-1,2,4-triazol-5-yl)-1H-indazole
4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}butan-1-one
1-(4-ethoxy-3-methylphenyl)-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
methyl 2-{[(4-fluorophenyl)methyl]sulfamoyl}-6-(3-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(2,3-dihydro-1H-isoindol-2-yl)-5,6,7,8-tetrahydroquinazolin-2-amine
N-(3-methylphenyl)-3-[1-(morpholine-2-carbonyl)piperidin-4-yl]propanamide
N-ethyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-(5-chloropyridin-2-yl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
4-[2-(5-acetylthiophen-3-yl)acetyl]-1λ6-thiomorpholine-1,1-dione
4-(2-methoxyquinolin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
2-amino-4-{3-[(dimethylamino)methyl]phenyl}-6-(5-methylpyridin-2-yl)pyridine-3-carbonitrile
4-ethoxy-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]pyrimidin-2-amine
1-(2,3-difluoro-4-methoxybenzoyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-{1-[(4-chlorophenyl)methyl]-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazol-3-yl}acetamide
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-1-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)ethan-1-one
1-(2-methoxyphenyl)-5-(oxolan-3-yl)-3-(propan-2-yl)-1H-1,2,4-triazole
5-{2-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-(2-methyl-1H-imidazol-1-yl)butanamide
1-[7-(1-benzothiophen-3-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
3-(2H-1,3-benzodioxol-5-yl)-1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
7-(2-methoxyethyl)-2-[3-(thiophen-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
7-[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-({6-[(1-methyl-5-oxopyrrolidin-3-yl)amino]pyrazin-2-yl}sulfanyl)acetic acid
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-4-methanesulfonyl-N-methylbenzamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}propanamide
3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)-1-[4-(piperidin-1-yl)piperidin-1-yl]propan-1-one
2-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-2-yl]pyridine
4-(2,3-dihydro-1H-inden-2-yl)-11-[ethyl(2-methylprop-2-en-1-yl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
5,6-dimethyl-3-[1-(pyrazin-2-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-{4-[(3-chloropyridin-4-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
2-ethyl-4-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1,3-oxazole-5-carboxamide
2-amino-4-{3-[2-(dimethylamino)ethoxy]phenyl}-6-(5-methylpyridin-2-yl)pyridine-3-carbonitrile
N-ethyl-N-(propan-2-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
3-{1-[1-(4-chlorophenyl)propan-2-yl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
2-[(4-chlorophenyl)methyl]-8-(2-propoxyacetyl)-2,8-diazaspiro[4.5]decan-3-one
1-(2-{[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}ethyl)imidazolidin-2-one
{[3-({1-[3-(4-fluorophenyl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl}(methyl)(thiophen-3-ylmethyl)amine
3-chloro-1-{2-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}-5-(trifluoromethyl)-1,2-dihydropyridin-2-one
5-(2,3,4,9-tetrahydro-1H-carbazole-7-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[(6-methylpyridin-2-yl)methyl]amine
2-(3-methylbutyl)-8-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1'-[(2-fluoro-5-methoxyphenyl)methyl]-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-4-(4-methylphenoxy)piperidine-4-carboxamide
(2R)-2-{[2-(cyclopropylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}-3-phenylpropan-1-ol
2-({4-[3-(hydroxymethyl)-8-methylquinolin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
N-[(3S,4R)-1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-(furan-2-ylmethyl)-2-(methoxymethyl)-N,6-dimethyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3-carboxamide
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}pyridazine-3-carboxamide
1-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methylbut-2-en-1-one