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2-(2-methoxyethyl)-9-(quinolin-6-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{2-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
methyl 9-(cyclopentyloxy)-3-{[4-(diethylamino)phenyl]methyl}-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-methyl-1-(1-methylpiperidin-4-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
9-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-4-[4-(trifluoromethyl)pyridin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
(2S,4S)-1-benzyl-N-ethyl-4-[(naphthalen-2-ylmethyl)amino]pyrrolidine-2-carboxamide
1-(2-chlorophenyl)-4-(4-oxo-4-phenylbutyl)piperazin-2-one
4-ethyl-3-(piperidin-4-ylmethyl)-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[3-(2-methoxyphenoxy)azetidin-1-yl]pyrimidin-4-amine
1-[4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepan-1-yl]ethan-1-one
N-cyclopentyl-2-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)propanamide
5-methyl-4-(4-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
(3S,4R)-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
6-methoxy-4-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]acetamide
5-({[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}carbamoyl)thiophene-2-carboxylic acid
N,N-dimethyl-3-[5-(pyrrolidin-1-ylmethyl)pyridin-2-yl]aniline
1-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
3-[2-(4-fluorophenyl)ethyl]-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine
2-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-1,2,3,4-tetrahydroisoquinolin-4-ol
3-{5-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-4-amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(morpholin-4-yl)propanamide
2-[(1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
(4aS,8aR)-6-(2-cyclopropylacetyl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-N-[2-(pyridin-3-yl)ethyl]pyridin-2-amine
(4aS,8aS)-4a-hydroxy-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-decahydroisoquinoline-2-carboxamide
2-fluoro-5-(1-methyl-1H-pyrazol-4-yl)benzoic acid
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(2-methylprop-2-en-1-yl)propanamide
1-[5-(3-chloro-5-fluorophenyl)-1H-1,3-benzodiazol-2-yl]ethan-1-ol
(4aS,8aR)-1-(3-hydroxypropyl)-6-(1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(2,3-dimethoxyphenyl)acetic acid
(3-{2-[1-(4,6-dimethylpyridine-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,4-difluorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
(1S,5R)-6-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
7-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-N-[phenyl(pyridin-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
4-methoxy-N-({1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
1-{2-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
ethyl 1-(1-acetylpiperidin-4-yl)-3-[(3-chlorophenyl)methyl]piperidine-3-carboxylate
methyl 4-[6-amino-5-cyano-4-(pyridin-3-yl)pyridin-2-yl]-5-methylfuran-2-carboxylate
3-(2-ethyl-1H-imidazol-1-yl)-1-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}propan-1-one
1-cyclohexyl-4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidine
dimethyl({4-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1,3-thiazol-2-yl}methyl)amine
(3aS,6aS)-2-cyclohexyl-5-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid