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1-benzyl-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-2-carboxamide
2-(butylsulfanyl)-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}pyrimidine
2-[4-(4-methylphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
3-{1-[2-(dimethylamino)-2-(2-fluorophenyl)acetyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-[2-(2-fluorophenyl)-1-(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)ethyl]-N-methylthiophene-2-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-(4-phenylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(cyclohexylmethyl)-5-[(3-hydroxy-2,2-dimethylpropyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-(4-methylphenyl)-4-[4-(4-methylpiperazin-1-yl)pentanoyl]piperazin-2-one
3-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
N-(1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-4-yl)pyrimidin-2-amine
(3aR,6aR)-2-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide
4-methyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzene-1-sulfonamide
2-(methylsulfanyl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3,5-dichloro-4-methyl-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
N-ethyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]quinoline-6-carboxamide
4-{4-[(5-ethylpyridin-2-yl)methyl]piperazin-1-yl}-6-methyl-2-propylpyrimidine
(2S)-3-phenyl-2-({2-[(propan-2-yl)amino]pyrimidin-5-yl}formamido)propanamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(quinolin-2-ylmethyl)pyrrolidin-3-yl]acetamide
2-({4-[2,5-dioxo-4-(pyridin-2-yl)imidazolidin-4-yl]piperidin-1-yl}methyl)benzonitrile
4-(1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-1,2,3-triazol-4-yl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
3-ethyl-4-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)-1H-pyrazole-5-carboxamide
2-({methyl[(2-methylpyridin-4-yl)methyl]amino}methyl)quinolin-4-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-4-(pyridin-2-yl)pyrimidin-2-amine
4-{4-[3-(1-methoxyethyl)phenyl]-6-methylpyrimidin-2-yl}morpholine
1-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
4-[6-(trifluoromethyl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]pyridine
3-(aminomethyl)-4-[(1S)-1-phenylpropyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(4-fluorophenyl)-2-{3-[(4-fluoropiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
2-{5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-1-yl}acetamide
3-tert-butyl-4-(5-ethylfuran-2-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2,3,6-trimethyl-4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]quinoline
5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-(oxolan-2-ylmethyl)-N-propyl-1,2-oxazole-3-carboxamide
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
3-[(dimethylamino)methyl]-N-[(1-hydroxycyclohexyl)methyl]benzamide
4-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-(2,3-dihydro-1H-inden-2-yl)pyrrolidin-2-one
N-(2-methanesulfonamidoethyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-[(benzylamino)methyl]-4-(pyridin-3-yl)phenol
4-{methyl[(3-methyl-1H-indol-2-yl)methyl]amino}-N-(propan-2-yl)pyridine-2-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
2-(4-chlorophenyl)-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]morpholine
8-[2-(3-fluorophenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}aniline
6-(methylsulfanyl)-2-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)piperidin-2-one
3-amino-1-{3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}propan-1-one
[4-(5-chloro-2,3-dihydro-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol