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3-({[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}methyl)-1λ6-thiolane-1,1-dione
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
2-cyclopropanecarbonyl-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
6-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
N-ethyl-2-(2-phenylethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]-1,3-benzoxazole-5-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[2-(dimethylamino)-6-(trifluoromethyl)pyrimidin-4-yl]piperidin-3-yl]propan-1-ol
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(oxan-4-yl)piperidine-3-carboxamide
1-(6-hydroxypyrimidin-4-yl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepan-6-ol
N-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide
(3aS,6aS)-2-[3-cyano-6-(propan-2-yl)pyridin-2-yl]-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
3-(pyrrolidin-1-ylmethyl)-1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-3-ol
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)naphthalene-1-carboxamide
N-[4-({ethyl[(5-methylfuran-2-yl)methyl]carbamoyl}methoxy)phenyl]propanamide
N-ethyl-6-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-methylpyrimidin-5-yl)quinoline-4-carboxamide
6-(2-chlorophenyl)-N-cyclopropyl-8-oxo-7-(prop-2-en-1-yl)-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
4-chloro-1-methyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-pyrazole-3-carboxamide
4-(3-fluorophenoxy)-1-(1H-imidazol-4-ylmethyl)piperidine-4-carboxylic acid
5-{[2-(cyclopentyloxy)phenyl]methyl}-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-oxo-2-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(pyridin-4-yl)-7-(thiophene-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(4-fluorophenyl)-1-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2,3,6-tetrahydropyridine
4-acetyl-N-(3-cyclopentaneamido-2-methylphenyl)-1,4-diazepane-1-carboxamide
2-chloro-4-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)phenol
(2S)-N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-4-methylpentanamide
4-[2-(1-methyl-1H-indol-3-yl)acetyl]morpholine-2-carboxylic acid
2-[(3-{[(4-methoxyphenyl)methyl](prop-2-yn-1-yl)carbamoyl}phenyl)amino]acetic acid
1-[1-(furan-3-ylmethyl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-benzyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1,3-thiazole-4-carboxamide
N-{2-[5-(3-methyl-1H-pyrazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}acetamide
(2R)-3-methyl-2-({4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)butan-1-ol
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
2-(4-methoxyphenoxy)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
2-[1-(furan-3-ylmethyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-yl]ethan-1-ol
3-(2-fluorophenyl)-5-(propane-1-sulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-cyclopropyl-1-(methoxymethyl)-N-[(3-methylthiophen-2-yl)methyl]cyclobutane-1-carboxamide
N-[2-(dimethylamino)ethyl]-3-[1-(1-methoxypropan-2-yl)piperidin-4-yl]propanamide
2-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}-N-methylacetamide
N,N-dimethyl-2-[2-({[3-(1H-1,2,4-triazol-1-yl)propyl]carbamoyl}amino)phenyl]acetamide
(3-benzyl-1-{[4-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methanol
(2S,4S)-N,N-diethyl-4-(2-hydroxyacetamido)-1-(4-methylbenzoyl)pyrrolidine-2-carboxamide
1-{4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-4-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 1-[(3R,5S)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-5-[(diphenylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(3-{2-[1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
2-[2-(cyclohexylamino)pyrimidin-5-yl]-N,N,6-trimethylquinoline-4-carboxamide
4-(1-{2-[methyl(1-methylpiperidin-4-yl)amino]acetyl}piperidin-3-yl)benzoic acid
5-(5-methylfuran-2-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1,2,4-triazin-3-amine