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N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(2-hydroxyacetyl)piperidin-3-yl]propanamide
1-(isoquinolin-5-yl)-3-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]urea
5-[(1,3-benzothiazol-2-ylmethyl)amino]-N,N-dimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}-2-[2-(methylsulfanyl)phenyl]acetic acid
N5-cyclopentyl-N3-methyl-1-(3-methylbutyl)-4-oxo-N3-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2,3,6-trimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}quinoline-4-carboxamide
(2R)-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
4-phenoxy-1-(thiophen-2-ylmethyl)piperidine-4-carboxylic acid
2-[4-(5-phenylmethanesulfonamido-1H-pyrazol-1-yl)piperidin-1-yl]propanamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-{2-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
2-benzyl-4-[(2-fluoro-4-methoxyphenyl)methyl]morpholine
methyl 3-[(3S,4R)-4-(morpholin-4-yl)-1-[(4-phenylphenyl)methyl]piperidin-3-yl]propanoate
3-(2-ethoxyethyl)-1-[(2-fluorophenyl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
methyl 4-[4-(5-{[(2-chlorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]pentanoate
[(5-ethylpyridin-2-yl)methyl][(4-methanesulfonylphenyl)methyl]methylamine
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-[2-(propan-2-ylsulfanyl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-[3-(morpholin-4-yl)propyl]-5-(1,2-oxazolidine-2-carbonyl)piperidin-2-one
2-{2-[(4-ethyl-1,4-diazepan-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetic acid
1-(2-chloropyridin-3-yl)-3-{2-[cyclopentyl(methyl)amino]ethyl}-3-methylurea
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(4-methylphenyl)methyl]oxane-2-carboxamide
(1R,5R)-6-[2-(2,4-difluorophenyl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
(2R,3R,6R)-5-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-ethyl-3-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
3-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4H-chromen-4-one
N-[2-(dimethylamino)ethyl]-4-(2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-cyclopentyl-2-phenyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
4-[(3S,4R)-4-hydroxyoxolan-3-yl]-N-{4-[(methylcarbamoyl)methyl]phenyl}-1,4-diazepane-1-carboxamide
N3-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1,3-dicarboxamide
6-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
4-cyclobutyl-N,6-dimethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
3-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-5-(oxolan-2-yl)-1,2,4-oxadiazole
1-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-3-(thiophen-3-yl)propan-1-one
(1R,3S)-3-ethoxy-7-(1-methyl-1H-indole-4-carbonyl)-7-azaspiro[3.5]nonan-1-ol
3-phenyl-N-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
5-(azepan-1-yl)-1-(cyclohexylmethyl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]oxolane-2-carboxamide
methyl 5-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-5-oxopentanoate
(3S,4R)-3-methoxy-1-(1-methyl-1H-indazole-3-carbonyl)piperidin-4-amine
[(1-ethyl-1H-indol-5-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
6-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(4-methoxyphenyl)-6,6-dimethyl-N-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-(2-{1-[(4-fluorophenyl)methanesulfonyl]piperidin-2-yl}ethyl)morpholine
methyl (1S,3S,3aR,6aS)-5-benzyl-1-(hydroxymethyl)-3-(5-methylfuran-2-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(2,2-dimethyloxan-4-yl)-2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{1-[(2,6-dichloro-3-hydroxyphenyl)methyl]pyrrolidin-3-yl}acetic acid
2-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4,6-dimethylpyridine-3-carbonitrile