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1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(2-methoxyphenyl)propan-1-one
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-{[4-(propan-2-yl)phenyl]methyl}-1,2-oxazole-5-carboxamide
4-(1-butyl-1H-imidazol-2-yl)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]piperidine
N-{1-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
7-(cyclopropylmethyl)-6-(2,5-dimethylfuran-3-yl)-8-oxo-N-propyl-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-[2-(benzenesulfonyl)ethyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
(1S,5R)-6-(cyclobutylmethyl)-3-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 2-(azepane-1-sulfonyl)-6-butanoyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
8-chloro-2-methyl-4-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoline
methyl 3-(furan-2-amido)-1-(3-methylbutyl)-5-[(1-methylpiperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(4-amino-5-methylpyrimidin-2-yl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-1,2,5,6,7,8-hexahydroquinolin-2-one
1,9-dimethyl-4-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,4,9-triazaspiro[5.5]undecane
4-[3-(2-oxopiperidin-1-yl)propanoyl]-1-phenylpiperazin-2-one
(4aS,8aR)-6-[(2,3-difluorophenyl)methyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-[(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amino]ethan-1-ol
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-1,2,3-benzotriazole-5-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(2,3-difluorophenyl)methyl]piperidine-3-carboxamide
5-(methoxymethyl)-3-[2-(methylsulfanyl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
(2R,3R)-3-(4-benzyl-1H-1,2,3-triazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-({2-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]phenyl}methyl)-1,4-diazepan-5-one
N-[(3R,4S)-1-(1H-imidazol-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
N-[(3S,4R)-1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1,3-dimethyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)-1-benzofuran-7-carboxamide
4-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-3-ylmethyl)piperidin-3-ol
2-(dimethylamino)-2-(4-fluorophenyl)-N-[1-(4-fluorophenyl)piperidin-4-yl]acetamide
(1S,2S,9S)-N-(5-carbamoyl-2-fluorophenyl)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
(3S,4S)-1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
1-[(4-methylnaphthalen-1-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-[(2-methylpyridin-3-yl)oxy]-1-(3-phenylpropyl)piperidine-4-carboxylic acid
3-[2-(3,4-difluorophenyl)ethyl]-1-(1,3-thiazol-2-ylmethyl)piperidine
5-{[2-(2-oxopyrrolidin-1-yl)ethyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(thian-4-yl)pyrrolidine-2-carboxamide
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
2-(2-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}phenoxy)propanoic acid
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-3,5-dimethyl-1,2-oxazole-4-sulfonamide
N-ethyl-6-methoxy-3-methyl-N-[(5-methylfuran-2-yl)methyl]-1-benzofuran-2-carboxamide
1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-methyl-8-(4-methylpyridin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-(morpholin-4-yl)propan-1-one
1-(1,3-benzothiazole-6-carbonyl)-3-(hydroxymethyl)piperidin-3-ol
4-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
3-(4-fluorophenyl)-5-{[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1,2,4-oxadiazole
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1,4-diazepan-5-one
methyl (1S,3S,3aR,6aS)-5-methyl-3-(6-methylpyridin-2-yl)-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2,4-dichloro-3-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}phenol
4-[(3S)-3-aminopyrrolidine-1-carbonyl]-N-[3-(4H-1,2,4-triazol-4-yl)propyl]benzene-1-sulfonamide