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2-ethyl-5-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}pyrimidine
3-methyl-5-[2-(thiophen-2-yl)ethyl]-1H-1,2,4-triazole
[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl](methyl)(piperidin-3-ylmethyl)amine
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
N-{[7-(3-chlorothiophene-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide
2-{[(2,2-dimethyloxan-4-yl)methyl](methyl)amino}-N,2-dimethylpropanamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(4H-1,2,4-triazol-4-ylmethyl)benzene-1-sulfonamide
N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(trifluoromethyl)benzamide
7-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-2-oxa-7-azaspiro[4.5]decane
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-4-methylpiperidine-1-sulfonamide
methyl (1R,3S,3aR,6aS)-3-[3-(difluoromethoxy)phenyl]-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
6-(2-aminoethyl)-2-methyl-N-[(1R,2S)-2-phenylcyclopropyl]pyrimidin-4-amine
(3S,4S)-1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
2-amino-4-(5-chlorothiophen-2-yl)-6-cyclopropanecarbonyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(1,3-benzothiazol-2-ylmethyl)-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-methylacetamide
5-[3-(propoxymethyl)pyrrolidine-1-carbonyl]-3-propyl-1H-pyrazole
1-(4-methoxyphenyl)-4-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-3-yl}piperazine
8-[3-(2-fluorophenyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
ethyl 3-[(2-fluorophenyl)methyl]-1-(quinoxaline-6-carbonyl)piperidine-3-carboxylate
N-{3-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-3-oxopropyl}acetamide
(3S,4S)-4-(naphthalen-2-yl)-1-(1H-pyrazole-3-carbonyl)piperidin-3-ol
7-ethyl-2-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]-N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}acetamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2-methylphenyl)methyl]acetamide
ethyl 1-(benzenesulfonyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
5-(3-fluorophenoxymethyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-5-methylthiophene-2-carboxamide
2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxamide
5-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N,4-trimethylpyrimidin-2-amine
8-chloro-2-[2-(trifluoromethyl)morpholin-4-yl]quinoline
4-{1-[1-(2-phenylpropyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carbonyl}morpholine
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
N-[2-(furan-2-yl)ethyl]-3,6,7-trimethyl-1-benzofuran-2-carboxamide
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-3,4-dihydropyrimidin-4-one
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl][(1-phenyl-1H-pyrazol-5-yl)methyl]amine
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
6,7-dimethyl-2-({2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1H-1,3-benzodiazole
N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N-(2,4-dimethoxyphenyl)-2-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]acetamide
2-[2-(3-hydroxypiperidin-1-yl)ethyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(2-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}phenyl)-1H-pyrazole
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
3-(5-{[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyridine
5,6-dimethyl-2-oxo-N-{3-[(pyridin-3-yl)amino]propyl}-1,2-dihydropyridine-3-carboxamide
4-ethyl-1-methyl-3-{[1-(quinoxalin-2-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(3,5-dimethoxyphenoxymethyl)-3-(phenoxymethyl)-1,2,4-oxadiazole
4-(benzyloxy)-1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea