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1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methylurea
(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl](quinolin-2-ylmethyl)amine
1-(2,3-dihydro-1H-inden-2-yl)-N-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-amine
1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
methyl 1-[(3R,5S)-1-propyl-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-ethyl-N-(2-methylprop-2-en-1-yl)piperidine-4-carboxamide
1-(2,6-diethylphenyl)-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-pyrazole-5-carboxamide
(7S,9aR)-N-(3-fluorophenyl)-7-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-2-ylmethyl)-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}propanamide
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
N-(2-methanesulfonamidoethyl)-2-(phenylamino)pyrimidine-5-carboxamide
2-[3-methyl-5-(2,3,4,9-tetrahydro-1H-carbazol-6-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
{[2-(furan-2-yl)pyrimidin-5-yl]methyl}(methyl)(quinolin-5-ylmethyl)amine
4-[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
({2,5-dimethyl-3-[(3-methylpiperidin-1-yl)methyl]phenyl}methyl)(methyl)(pyrazin-2-ylmethyl)amine
3-(1-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(methylsulfanyl)propanamide
6-(4-{[2-(3-phenylpyrrolidin-1-yl)ethyl]amino}piperidin-1-yl)pyridine-3-carbonitrile
2-methoxy-N-{1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(2R,6R)-11-methoxy-4-(4-methyl-1H-imidazole-2-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
[(8-methoxy-2H-chromen-3-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
6-[(diethylamino)methyl]-N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
(2S,4S)-4-{[(3-methylphenyl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazine-1-carbonyl]-1,4-dihydroquinolin-4-one
2-[3-(3,4,5-trimethoxyphenyl)phenyl]ethan-1-amine
1-(cyclohexylmethyl)-5-[(5-hydroxyadamantan-2-yl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-(hydroxymethyl)piperidin-3-ol
3-[1-(1-methylpiperidin-4-yl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide
7-methoxy-3-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1H-3-benzazepine
1-[5-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)-1-methyl-1H-pyrrol-3-yl]ethan-1-one
N-{[7-(1H-indole-6-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-3-yl)acetamide
(2S,4S)-4-amino-N-[(4-ethylphenyl)methyl]-N-[(2-methoxyphenyl)methyl]-1-methylpyrrolidine-2-carboxamide
methyl 1-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]piperidine-4-carboxylate
N-methyl-N-{4-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]phenyl}methanesulfonamide
N-ethyl-5-(2-fluorophenoxymethyl)-N-(2-hydroxyethyl)-1H-pyrazole-3-carboxamide
2-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
(4aS,7aR)-1-(5-oxo-2,5-dihydro-1H-pyrazole-3-carbonyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(5-oxo-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
(2-{2-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
2-(4-chlorophenyl)-4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]morpholine
N-(4-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}phenyl)acetamide
(3S,4R)-4-methyl-1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidine-3,4-diol
N-(3,4-dimethoxyphenyl)-1-[1-(2-methylphenyl)piperidin-4-yl]piperidin-3-amine
1-(furan-3-ylmethyl)-5-(4-methanesulfonylphenyl)-4-phenyl-1H-imidazole
3,4-dimethoxy-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
2-cyano-N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
4-(dimethylamino)-N,N-dimethyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-sulfonamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-4-(piperidin-1-ylmethyl)benzamide
N-(4-{methyl[1-(methylcarbamoyl)propan-2-yl]carbamoyl}phenyl)pentanamide