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methyl 2-(azocane-1-sulfonyl)-6-(2,2-dimethylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(6-methoxynaphthalen-2-yl)morpholine
3-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}-2-chloro-6-methoxyphenol
5-acetyl-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4,4,4-trifluoro-1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}butan-1-one
6-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}-2-(1H-indol-3-yl)acetamide
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]ethan-1-one
5-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrole-2-carbonyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine
5-ethyl-N4-[3-(pyridin-3-yl)propyl]pyrimidine-2,4-diamine
N-(cyclohexylmethyl)-2-[(3S,4R)-3-cyclopropyl-4-acetamidopyrrolidin-1-yl]acetamide
(4S)-3-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-(propan-2-yl)-1,3-oxazolidin-2-one
5-cyclopropyl-N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-1H-pyrazole-3-carboxamide
4-[(dimethylamino)methyl]-1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}azepan-4-ol
1-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-2-(2-ethoxyphenyl)-1H-imidazole
4-(5-fluoro-1,3-dimethyl-1H-indole-2-carbonyl)-3-(4-fluorophenyl)piperazin-2-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylacetamide
6-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoxaline
N-(1-methylpiperidin-4-yl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[2-(4-{[3-(3,4-dimethoxyphenyl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]cyclobutanecarboxamide
3-{[(4-phenyl-1,3-thiazol-2-yl)methyl](pyridin-4-ylmethyl)amino}propan-1-ol
[(1-cyclohexylpiperidin-3-yl)methyl][(3-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(3-methoxyphenyl)azetidin-1-yl]ethan-1-one
2-hydroxy-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]butanamide
1-[(4-fluorophenyl)methyl]-4-(2-methoxypyridine-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
8-cyclopropanecarbonyl-2-[(4,5-dimethylfuran-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(piperazin-1-yl)-2-[3-(1H-pyrazol-1-yl)propyl]-2,3-dihydropyridazin-3-one
1-(4-methoxybenzoyl)-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}piperazine
5-{furo[3,2-c]pyridin-4-yl}-1,2,3,4-tetrahydroisoquinoline
5-acetyl-6-methyl-2-oxo-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1,2-dihydropyridine-3-carboxamide
(3S,4S)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
2-(methylsulfanyl)-5-({3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyrimidine
1-(4-benzylpiperidin-1-yl)-3-[1-(6-methylpyridine-3-carbonyl)piperidin-4-yl]propan-1-one
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-6-(trifluoromethyl)pyridine-3-carboxamide
1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}ethan-1-one
N-methyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
N-[1-(dimethylamino)propan-2-yl]-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(4-{[1-(dimethylamino)butan-2-yl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazin-1-yl]propan-1-one
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methyl-2-(naphthalen-2-yloxy)propanamide
3-{1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
{3-[(2,4-difluorophenyl)methyl]-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-yl}methanol
5-acetyl-3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}acetic acid
N-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-[(2-chloro-4-fluorophenyl)methyl]azonan-2-one
8-(3-fluoropyridin-2-yl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-cyclopropylpyrimidine
1-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-methyl-3-(morpholin-4-yl)propan-1-one
ethyl 5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate