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4-({2-[1-(4-fluoro-3-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(methoxymethyl)-N-methylcyclopropan-1-amine
N-tert-butyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-5-[(2-phenylpropyl)amino]benzene-1-sulfonamide
6-(2-fluoro-6-methoxyphenyl)-N-(propan-2-yl)pyrimidin-4-amine
1-(4-chloro-2-fluorophenyl)-3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-methylurea
3-[1-(but-2-ynoyl)piperidin-3-yl]-N-[(3,4-difluorophenyl)methyl]propanamide
ethyl 4-[(2-methyl-1-benzofuran-5-yl)carbamoyl]piperazine-1-carboxylate
1-methyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carboxamide
5-[1-(furan-2-carbonyl)pyrrolidin-2-yl]-N-[2-(1H-imidazol-4-yl)ethyl]thiophene-2-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}ethan-1-one
1-[(4-chlorophenyl)methyl]-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)piperidin-2-one
(3R,4R)-N-[(3-fluorophenyl)methyl]-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carboxamide
1-(3,5-dimethylphenyl)-3-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
3-(2,6-dimethylpyridin-3-yl)-1-methyl-1-[1-(pyrimidin-4-yl)ethyl]urea
N-{[1-(2,2-dimethylpent-4-en-1-yl)piperidin-3-yl]methyl}acetamide
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-(2-cyclopropylacetyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-(1,4-dioxan-2-ylmethyl)-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(3R,4R)-1-(2,3-difluorobenzoyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
1-(2,1,3-benzothiadiazol-5-ylmethyl)-1-methyl-3-[3-methyl-1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
1-cycloheptyl-4-[(1H-imidazol-4-ylmethyl)amino]pyrrolidin-2-one
N,1,3-trimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-butyl-8-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-methyl-1-[2-(morpholin-4-yl)ethyl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
N-[4-(pyridin-3-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyridazine-3-carboxamide
1-[3-(1,2-oxazol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-phenoxypropan-1-one
2-[2-methoxy-1-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]pyridine
ethyl 1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-imidazole-2-carboxylate
6-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-6-benzyl-3-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(2,6-dimethylpyridin-4-yl)piperazine
2-(2-chlorophenyl)-3-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(4-cyclohexyl-3-oxopiperazine-1-carbonyl)-3,4-dihydroquinazolin-4-one
2,3-dimethyl-6-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}quinoxaline
8-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-propyl-1,3,4-thiadiazol-2-amine
(2S,4S)-4-amino-N,N-diethyl-1-(9H-fluorene-9-carbonyl)pyrrolidine-2-carboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
3-{2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-5-hydroxy-4-oxo-4H-pyran-2-carboxamide
[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
N-[(3-methylphenyl)methyl]-4-(1H-pyrazol-4-yl)butanamide
5-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-propyl-1,2,4-oxadiazole
1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-(2-methoxyphenoxy)-1-(pyrazin-2-yl)piperidine-4-carboxylic acid
5-{2-amino-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}-1-propylpiperidin-2-one
5-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-3,4-dihydropyrimidin-4-one
2-[2-(2-amino-3-cyano-5-methyl-6-phenylpyridin-4-yl)phenoxy]acetic acid