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2-[1-(quinoline-5-carbonyl)pyrrolidin-3-yl]benzoic acid
4-(3,5-dimethylfuran-2-carbonyl)-2-[(3-methoxyphenyl)methyl]morpholine
2-methoxyethyl 2-(3-methoxyphenyl)piperidine-1-carboxylate
1-({3-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-indole
3-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]-5-(thiomorpholine-4-sulfonyl)benzoic acid
4-[(3-fluorophenyl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
4-(1-tert-butyl-1H-pyrazol-4-yl)-1-[2-(piperidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridine
2-(pyridin-4-ylmethyl)-8-[2-(pyrrolidin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-amino-4-(1,5-dimethyl-1H-pyrazol-4-yl)-5-methyl-6-phenylpyridine-3-carbonitrile
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
(furan-2-ylmethyl)[(4-methanesulfonylphenyl)methyl](thiophen-3-ylmethyl)amine
7-(1H-pyrazol-3-yl)-3,4-dihydro-2H-1-benzopyran-4-one
5-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
ethyl({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-3-methyl-1-propyl-1H-pyrazole
[2-(1H-imidazol-1-yl)ethyl](methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
(1S,5R)-3-{[2-(benzylamino)pyrimidin-5-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,4S)-2-(2-fluorophenyl)-5-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)-2-(pyridin-3-yloxy)acetamide
N,N-dimethyl-5-({4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridin-2-amine
4-chloro-N,N-dimethyl-5-[1-(pyridin-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,3-thiazol-2-amine
N5-(pyridin-3-ylmethyl)-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[2-hydroxy-3-(4-methoxy-2-{[methyl(oxan-4-yl)amino]methyl}phenoxy)propyl]piperidin-4-ol
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-[(2-chlorophenyl)methyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-chlorophenyl)-3-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}propanamide
4-{1-[(4-methanesulfonylphenyl)methyl]piperidin-4-yl}pyridine
2-[(1S,5R)-3-(3-cyano-4,6-dimethylpyridin-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
1-(carbamoylmethyl)-N-cyclopentyl-N-(prop-2-en-1-yl)piperidine-3-carboxamide
1'-[2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
3,3-dimethyl-1-[2-(propan-2-ylsulfanyl)phenyl]urea
3-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-1λ6-thiane-1,1-dione
N-[(3S,4R)-4-(4-methylphenyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]cyclopropanecarboxamide
6-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-{1-[4-(1H-imidazol-1-yl)benzoyl]pyrrolidin-2-yl}-N,N-dimethylthiophene-2-carboxamide
[1-(5-phenyl-1H-pyrrole-2-carbonyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
2-(2-methoxyethyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}-4-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}piperazine
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-4-hydroxy-2-(phenoxymethyl)pyrimidine-5-carboxamide
8-methyl-3-(3-phenoxyazetidine-1-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane
2-({[(3-cyanophenyl)carbamoyl]amino}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-4-(piperidin-1-yl)piperidine-4-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(pyridin-3-yloxy)ethyl]-1H-pyrazole-4-carboxamide
N-(pyridin-3-ylmethyl)-3-{1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-4-yl}propanamide
3-[5-(3,3-dimethylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(2-hydroxyethyl)propanamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(1H-pyrazol-1-yl)benzamide