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(4aS,7aR)-1-(1-aminocyclopropanecarbonyl)-4-cyclobutanecarbonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
N-(1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidin-3-yl)acetamide
1-{6-[(3,5-dimethoxyphenyl)methoxy]-3-oxo-4-(propan-2-yl)-1,4-diazepan-1-yl}-2-phenylethane-1,2-dione
[(3R,4R)-1-(4-fluorobenzoyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
2-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)pyridine-3-carbonitrile
6-{[4-(thiomorpholine-4-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
5,6-dimethyl-N-[1-(5-methylpyridin-2-yl)propyl]pyrimidin-4-amine
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(oxan-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-2-(2,3-dihydro-1H-inden-1-yl)acetamide
6-methyl-2-(3-phenoxypropyl)pyridine-3-carbonitrile
7-[1-(4-chlorophenyl)cyclobutanecarbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
{1-[4-(1H-indol-3-yl)butan-2-yl]-4-[(3-methoxyphenyl)methyl]piperidin-4-yl}methanol
N-cyclopropyl-1-methyl-N-(naphthalen-1-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperazin-2-one
2-(1-{1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidin-3-yl}-N-methylformamido)-N-methylacetamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)but-3-enamide
2-(4-fluorophenoxymethyl)-4-hydroxy-N-methyl-N-[(2-methylpyridin-4-yl)methyl]pyrimidine-5-carboxamide
6-[(diethylamino)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(ethylamino)-4-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1,3-thiazole-5-carboxamide
N-[(1,4-dimethylpiperazin-2-yl)methyl]-3-(3-hydroxyphenyl)propanamide
5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(2-methoxyphenyl)-1,2,4-oxadiazole
3-{[(2-hydroxy-2-phenylethyl)(methyl)amino]methyl}-7-methyl-1-[(3-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
4-methyl-2-(4-methylpiperazin-1-yl)-N-[(5-methylpyrazin-2-yl)methyl]pyrimidine-5-carboxamide
N-[3-({[2-(1H-imidazol-1-yl)propyl]carbamoyl}amino)phenyl]butanamide
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-1-propyl-1H-1,2,3-triazol-4-amine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-(piperidin-1-yl)cyclohexane-1-carboxamide
(3S)-3-ethyl-4-[1-(oxan-4-yl)piperidine-4-carbonyl]morpholine
3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
(butan-2-yl)[(6-methylpyridin-2-yl)methyl](thiophen-3-ylmethyl)amine
(1S,3R)-3-amino-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]cyclopentane-1-carboxamide
(1S,5R)-3-benzyl-6-(4-chloro-3-methylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-[(3-methoxyphenyl)methyl]-4-(3-methylfuran-2-carbonyl)-1,4-diazepan-2-one
4-[(3-methoxypropyl)amino]-5-methyl-N-(3-methylbutyl)thieno[2,3-d]pyrimidine-6-carboxamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-methyl-7-{4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanoyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
5-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-({ethyl[2-hydroxy-2-(3-hydroxyphenyl)ethyl]amino}methyl)-8-methyl-1,2-dihydroquinolin-2-one
4-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-1-phenylpiperidine
methyl 6-[(2,5-dimethylphenyl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N,N-dimethyl-3-[methyl(oxan-2-ylmethyl)sulfamoyl]benzamide
2-(3-chloro-4-hydroxyphenyl)-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}ethan-1-one
1-(5-chloropyridin-2-yl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylic acid
1-{[3-(4-ethenylphenoxy)-4-methoxyphenyl]methyl}pyrrolidine
2-(3-{3-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)acetamide
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-{[(4-fluorophenyl)methyl](methyl)amino}ethan-1-one
2-[5-benzyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
2-(dimethyl-1,3-thiazol-5-yl)-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[2-(ethanesulfonyl)ethyl]-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one