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11-[(3-ethoxypropyl)amino]-4-[2-(4-methoxyphenyl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N,6-dimethyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-(1,4-dioxane-2-carbonyl)-4-(pyridin-3-ylmethyl)piperazine
2-[(1S,5R)-3-(3-fluoropyridin-2-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-(dimethyl-1,3-thiazole-4-carbonyl)-4-azatricyclo[4.3.1.13,8]undecane
3-[(dimethylamino)methyl]-1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-ol
2-hydroxy-3-(2-methylphenoxy)-N-[2-(1,3-thiazol-4-yl)ethyl]propanamide
4-{5-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
5-{[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzothiadiazole
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-[2-(1,3-thiazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-(pyridin-2-ylmethyl)-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-[4-(methylsulfanyl)phenyl]acetamide
2-[2,4-dioxo-1-(2-phenylethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
5,5-dimethyl-3-(2-{2-methyl-4-[(3-methylphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1,3-oxazolidine-2,4-dione
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
N-(2-hydroxyethyl)-2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
8-(2-amino-2-methylpropyl)-3-{2-[methyl(2-phenylethyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5,6-dimethoxy-2-(2-{6-oxa-9-azaspiro[4.5]decan-9-yl}-2-oxoethyl)-1,2-dihydroisoquinolin-1-one
(1S,5R)-6-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
3-[3-({[(4-methylphenyl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
3-(3,5-dimethylphenyl)-N-[(5-methylpyrazin-2-yl)methyl]propanamide
1-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
4-{5-[(4-benzylpiperidin-1-yl)methyl]-1,3-thiazol-2-yl}morpholine
7-methoxy-1-methyl-2-[2-(1H-1,2,4-triazol-3-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
4-[5-(3-methoxyphenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
1-[4-(adamantan-1-yl)piperazin-1-yl]-2-(1H-pyrazol-1-yl)propan-1-one
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-methyl-N-[1-({2-oxo-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-3-yl}methyl)pyrrolidin-3-yl]acetamide
methyl({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(pyrazin-2-ylmethyl)amine
4-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydroisoquinolin-1-one
1-(2-chloroprop-2-en-1-yl)-7-fluoro-3-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
3-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(5-methanesulfonamido-2-methylphenyl)urea
methyl 5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
3-methoxy-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}pyridine-2-carboxamide
4-(hydroxymethyl)-3-{[2-(trifluoromethyl)phenyl]methyl}-1,3-oxazolidin-2-one
2-(6-methoxypyridin-3-yl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-(1H-1,2,4-triazol-3-ylsulfanyl)ethan-1-one
5,7-dimethyl-N-[4-(pyrrolidin-1-yl)butyl]pyrido[2,3-d]pyrimidin-4-amine
3-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
(3R,4R)-1-(4-chloro-2-methoxybenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-{[4-(2-methoxyethoxy)phenyl]methyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-hydroxy-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)benzamide
1-methyl-8-[3-(5-methylfuran-2-yl)butyl]-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1-methyl-1H-pyrazole-5-carboxamide
8-[(2R)-2-aminopropanoyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
1-{[2-(cyclopentyloxy)phenyl]methyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-[1-(furan-2-yl)ethyl]-5-methyl-1H-pyrazole-4-carboxamide