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(2S,3R)-2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)-3-hydroxybutanamide
7-fluoro-3-methyl-2-[4-(2-phenoxyethyl)piperazine-1-carbonyl]-1H-indole
N-[2-(dimethylsulfamoyl)ethyl]-4-oxo-4H-chromene-2-carboxamide
2,6-dimethoxy-N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)pyrimidine-4-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-(1,2-oxazinan-2-yl)ethan-1-one
6-(methoxymethyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}pyrimidin-4-amine
(1S)-3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-phenylpropan-1-ol
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
[(3R,4R)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
1-[2-(dimethylamino)ethyl]-5-oxo-N-{2-[2-(trifluoromethyl)phenyl]ethyl}pyrrolidine-3-carboxamide
1-[4-({4-[(2-chloro-6-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
1-(cyclopropylmethyl)-5-(quinolin-4-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-methoxy-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-(2-hydroxyethyl)-1-methyl-N-(1,3-thiazol-2-ylmethyl)azepane-2-carboxamide
3-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-N-phenylpropanamide
4-[5-(3-ethoxybenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]-1H-pyrazole
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-[(4-phenylphenyl)methyl]pyrrolidin-3-yl]methanol
N-[2-(4-chlorophenyl)ethyl]-2-{[2-(1H-imidazol-4-yl)ethyl]amino}acetamide
9-[4-(1,3-oxazol-5-yl)benzenesulfonyl]-3,9-diazaspiro[5.6]dodecane
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-(pyrimidin-2-yl)-1H-pyrazol-1-yl]acetamide
methyl 3-(butanamidomethyl)-5-[1-(4-chlorophenyl)cyclopropaneamido]benzoate
3-chloro-4-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-[2-(dimethylamino)ethyl]benzamide
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-(4-methylphenyl)-4-[2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperazin-2-one
(2R)-2-hydroxy-N-methyl-N-[(4-phenoxyphenyl)methyl]propanamide
N-{1-[(4-fluorophenyl)methyl]-7-(3-oxopiperazine-1-carbonyl)-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
6-ethyl-2-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-dihydropyridine-4-carboxamide
1-[(3-methyl-1H-indol-2-yl)methyl]-4-phenoxypiperidine-4-carboxylic acid
3-[(3,4-dimethoxyphenyl)methyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-(propylsulfanyl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
4-(2-chlorophenoxy)-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]piperidine
2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3-phenylpropanamide
N-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
(1S,5R)-3-methyl-6-(3,4,7-trimethyl-1H-indole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
N-[2-(2-fluorophenyl)ethyl]-5-{4-hydroxy-1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
4-(2,6-dimethoxypyridine-3-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
1-methyl-4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidine
1-[(2-chlorophenyl)methyl]-7-fluoro-3-({[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-[1-(pyridin-2-yl)propyl]acetamide
8-[3-(1H-imidazol-2-yl)benzoyl]-1-oxa-8-azaspiro[4.5]decane
N-(3-chloro-4-fluorophenyl)-3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
3-(1H-1,3-benzodiazol-1-yl)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
5-acetyl-6-methyl-2-oxo-N-[2-(phenylsulfanyl)ethyl]-N-(prop-2-en-1-yl)-1,2-dihydropyridine-3-carboxamide
4-cyano-N-({1-[(1-ethenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
1-(4-methoxyphenyl)-4-(2-methyloxane-2-carbonyl)piperazin-2-one
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-4-(2-methylpropyl)pyrrolidin-2-one