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N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
3-methyl-N-{2-methyl-3-[(1,3-thiazol-2-yl)carbamoyl]phenyl}-1H-pyrazole-5-carboxamide
5-(3,6-dimethylpyrazin-2-yl)-1H-indole
2-methoxy-N-(1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(3S,5R)-N3-cyclohexyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]piperidine-3,5-dicarboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-(oxolan-3-ylmethyl)piperidine-4-carboxamide
2-{5-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
4-amino-N-(2-benzamido-5-methylphenyl)pyridine-2-carboxamide
4-{[4-(methylsulfanyl)phenyl]methyl}-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-benzyl-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-oxopyrrolidine-3-carboxylic acid
4-(hydroxymethyl)-1-{[5-(pyridin-2-yl)thiophen-2-yl]sulfonyl}piperidin-4-ol
1-(1-cyclohexanecarbonylpiperidin-4-yl)-N-cyclopropylpiperidine-3-carboxamide
8-fluoro-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)quinoline-2-carboxamide
N-cyclopropyl-3-phenyl-N-(3-phenylprop-2-yn-1-yl)-1H-pyrazole-4-carboxamide
(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-7-({[3-(methylsulfanyl)phenyl]methyl}amino)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[benzyl(methyl)amino]-N-(1-hydroxy-2-methylpropan-2-yl)-2,3-dihydro-1H-indene-2-carboxamide
1-cyclohexyl-N-methyl-4-oxo-5-(4-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
3-[1-(6-aminopyridin-2-yl)-4,5-dimethyl-1H-1,3-benzodiazol-2-yl]propanoic acid
N-{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}-2,2-dimethyloxan-4-amine
4-{[(3R,4S)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]methyl}benzamide
4-[2-(dimethylamino)benzoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
ethyl 3-benzyl-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-3-carboxylate
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-{[4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
1-[(3-fluorophenyl)methyl]-4-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperazin-2-one
{5-[1-(1-benzylpyrrolidin-3-yl)-1H-imidazol-2-yl]furan-2-yl}methanol
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-(2-hydroxyethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
1-{1'-[6-(dimethylamino)pyrazin-2-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
8-(2-methoxyethyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
8-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(3-phenylpropyl)-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1,4-diazepane
[4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]methanamine
5-fluoro-2-(4-{[3-(4-fluorophenyl)morpholin-4-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
N,N-dimethyl-2-(1,4-oxazepan-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-sulfonamide
{[4-methoxy-3-(methoxymethyl)phenyl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-cyclohexyl-N-(2-phenylethyl)-2-(pyrrolidin-3-yl)acetamide
2-(2,5-dimethoxyphenyl)-1-[3-(2-methylphenoxy)azetidin-1-yl]ethan-1-one
N-cyclopentyl-5-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-1-benzoxepine-4-carboxamide
2-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile
N-[2-(1-benzyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-3-methoxybenzamide