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(1S,5R)-6-(cyclopropylmethyl)-3-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[1-(hydroxymethyl)cyclopentyl]acetamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-{1-[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
5-(methoxymethyl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)furan-2-carboxamide
5-acetyl-N-[3-(azepan-1-yl)propyl]-N-methylthiophene-3-carboxamide
3-[(dimethylamino)methyl]-1-(2,2-diphenylethyl)pyrrolidin-3-ol
1-methyl-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
(3R,4R)-1-{[4-(benzyloxy)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
4-benzyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-one
N-[3-(3,4-dimethoxyphenyl)propyl]-5-methylpyrimidin-2-amine
N,N-dimethyl-5-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}pyrimidin-2-amine
N-(3-{4-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]piperidin-1-yl}phenyl)-2-methoxybenzamide
methyl (2S,4R)-1-[(4-fluorophenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
1-{1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
11-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-cyclohexyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidine-4-carboxamide
N-(prop-2-en-1-yl)-7-{pyrazolo[1,5-a]pyridine-3-carbonyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(4-methoxy-3-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}phenyl)-4H-1,2,4-triazole
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[1-(pyridin-3-yl)propan-2-yl]propanamide
6-(1H-1,3-benzodiazol-1-yl)-2H-1,3-benzodioxole-5-carboxamide
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-[(dimethylamino)methyl]piperidin-3-ol
2-[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]-3-phenylpropanoic acid
N'-(2,3-dimethylphenyl)-N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}propanediamide
N-{2-[methyl(2-phenylethyl)amino]ethyl}-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
({3-[(1-cyclohexanecarbonylpiperidin-3-yl)methoxy]phenyl}methyl)(methyl)(quinolin-6-ylmethyl)amine
(2S,4R)-4-amino-N,N-diethyl-1-[2-(4-fluoro-3-methylphenyl)acetyl]pyrrolidine-2-carboxamide
1-[(3,4-difluorophenyl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-{3-[(3,4-dimethoxyphenyl)methyl]-5-methyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
methyl 3-[({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)(oxolan-2-ylmethyl)sulfamoyl]thiophene-2-carboxylate
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(4-fluorophenoxy)ethan-1-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}propan-1-one
7-cyclohexyl-2-[3-(pyridin-2-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
8-(1-methoxypropan-2-yl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 5-[(1-ethylpiperidin-4-yl)amino]-1-[2-(1H-indol-3-yl)ethyl]-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-tert-butyl-1-cyclohexyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
(1S,3R)-3-amino-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]cyclopentane-1-carboxamide
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-({1-[(4-methylphenyl)methyl]-3-phenyl-1H-1,2,4-triazol-5-yl}methyl)morpholine
4-(3-benzyl-1H-pyrazol-5-yl)-1-(piperidin-3-yl)piperidine
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
5-[2-(naphthalen-1-ylmethyl)morpholine-4-carbonyl]pyridin-2-ol
6-chloro-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-1,3-benzothiazol-2-amine
(1R,5R)-3-(2,3-dimethoxybenzoyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
(3S)-3-benzyl-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-2-one
3-{[1-(3-cyanopyridin-2-yl)pyrrolidin-3-yl]methyl}benzoic acid
1-[5-methoxy-2-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-(cyclobutylmethyl)-4-oxo-N-(oxolan-2-ylmethyl)-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-phenoxyethyl)piperazine