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N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carboxamide
11-[(prop-2-en-1-yl)amino]-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N4-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5-ethyl-6-methylpyrimidine-2,4-diamine
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(3-methylphenoxy)ethan-1-one
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(pyridin-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylcyclohex-1-ene-1-carboxamide
2-({5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}amino)ethan-1-ol
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(1-methylpiperidin-2-yl)propan-1-one
N'-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,N,N'-trimethylbutanediamide
N-{2-[5-(1-ethyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridin-3-amine
4-[(2,3-difluorophenyl)methyl]-3-{2-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
5-methanesulfonyl-N-methyl-N-(3-phenylpropyl)-4-(piperidin-3-yl)pyrimidin-2-amine
N-(2-hydroxy-3-methoxypropyl)-N-methyl-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
N-[(5-chloro-2,3-dimethoxyphenyl)methyl]-1-(methoxymethyl)-N-methylcyclopropan-1-amine
2-[1-(cyclohexylmethyl)-4-(thian-4-yl)piperazin-2-yl]ethan-1-ol
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
3-ethyl-1-{2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carbonyl}piperidin-3-ol
dimethyl({4-methyl-5-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-(4-methylpiperazin-1-yl)benzamide
4-ethyl-1-methyl-3-({1-[2-(pyridin-3-yloxy)acetyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(4-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-[(2E)-2-methylbut-2-en-1-yl]-7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[2-(1H-indol-3-yl)ethyl]-3-pentanamidobenzamide
(1S,5R)-N-(2-methylphenyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
4-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}pyridine
ethyl 4-{3-azaspiro[5.5]undecan-9-yl}piperazine-1-carboxylate
3-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]benzonitrile
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-{2-ethyl-4-[2-(hydroxymethyl)phenyl]phenyl}acetamide
1-{[(2R,5S)-5-(naphthalen-1-ylmethyl)oxolan-2-yl]methyl}piperidine-4-carboxylic acid
1-(5-methanesulfonyl-2-methylphenyl)-3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]urea
3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-1-(thiophene-2-carbonyl)piperidine
5-cyclobutanecarbonyl-1'-(2-methyl-1H-pyrrole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2-methyl-3-phenylcycloprop-2-ene-1-carbonyl)piperidine
N-[2-(furan-2-yl)ethyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
5,7-dimethyl-N-[2-(piperidin-1-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
1-(2-cyclohexylethyl)-3-hydroxy-3-{[(propan-2-yl)amino]methyl}piperidin-2-one
N-[(3R,4S)-1-(5-ethyl-2-methylpyrimidin-4-yl)-4-propylpyrrolidin-3-yl]methanesulfonamide
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-({1-[6-(butylamino)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
(2R,3R)-3-[4-(2-ethoxyethyl)piperazin-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(naphthalen-2-ylmethyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclopropyl-1-[2-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-[(3S,4R)-1-benzyl-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(pyridin-2-ylmethyl)propanamide
3,6-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-[5-(4-methoxyphenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide