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2-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrrole
2-[(5-methylpyrazin-2-yl)methyl]-8-[(5-methylthiophen-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(pyrimidin-4-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-4-(pyridin-3-yl)piperidin-4-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}propanamide
1-({[1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-yl]amino}methyl)cyclohexan-1-ol
(3S,4S)-4-methyl-1-[2-(6-methylpyridin-2-yl)ethyl]piperidine-3,4-diol
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
5-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-pyrazol-3-yl]-4-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazol-2-amine
N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-4-(trifluoromethyl)benzamide
1-(4-methylphenyl)-4-(2-phenylbutanoyl)piperazin-2-one
7-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-phenyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-1,2,4-triazin-3-amine
4-{1-[(4-chlorophenyl)methyl]pyrrolidin-3-yl}-1-methanesulfonylpiperidine
2-{2-cyclobutanecarbonyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1-methyl-1H-1,3-benzodiazole
3-(2-methylphenyl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]propanamide
2,3-dimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}pyrrolidin-2-yl)pyridine
N-methyl-N-(quinolin-5-ylmethyl)-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
5-[1-(2H-1,3-benzodioxol-5-yloxy)ethyl]-3-cyclopropyl-1H-1,2,4-triazole
5-{[2-(dimethylamino)-2-(3-fluorophenyl)acetamido]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
2-chloro-4-{[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]methyl}-6-methoxyphenol
1-[6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridin-3-yl]ethan-1-one
4-{5-[(2,5-dimethoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}morpholine
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1-cyclohexylpiperazin-2-yl]ethan-1-ol
5-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methoxypyrimidine
5-(2,2-dimethylpropanoyl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{1-[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]-2-phenylethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
dimethyl[(5-{[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}thiophen-3-yl)methyl]amine
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
8-cyclopropanecarbonyl-2-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[2-(4-acetylpiperazin-1-yl)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)cyclohexanecarboxamide
3-(2-fluoroethyl)-5-(3-phenylpropyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-(3,5-dimethylphenyl)-4-[(2R)-pyrrolidine-2-carbonyl]piperazin-2-one
3,3-dimethyl-4-(4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanoyl)piperazin-2-one
(1S,5R)-3-({2-ethyl-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl}methyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({7-[2-(2-chloro-4-fluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-2-carboxamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2,5,6-trimethylpyrimidin-4-amine
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-methyl-N-[(5-methylfuran-2-yl)methyl]-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}morpholine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(propane-1-sulfonyl)piperidin-3-yl]piperazine
2-amino-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-5-methyl-6-(thiophen-2-yl)pyridine-3-carbonitrile
(2S,4S)-4-[(adamantan-2-yl)amino]-1-[(2-chlorophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
(3S,4S)-1-{[2-(cyclopentyloxy)phenyl]methyl}-4-(dimethylamino)pyrrolidin-3-ol
1-{4-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]-6-hydroxy-1,4-diazepan-1-yl}ethan-1-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(furan-3-ylmethyl)-N-methylpyrimidin-2-amine
[(3aS,6aS)-2-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
4-methoxy-N-(2-methoxyethyl)-2-{[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]oxy}benzamide