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2-methyl-5-{2-[2-({5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}amino)ethyl]morpholin-4-yl}-2,3-dihydropyridazin-3-one
N-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-4-(2-phenoxyethyl)piperazine-1-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-hydroxy-N,3-dimethylbenzamide
N-[1-(3,4-dimethoxyphenyl)ethyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-[3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazole
3-{[4-(2-amino-6-methylpyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]methyl}benzonitrile
(2R,6S)-2,6-dimethyl-4-[1-(1-methyl-1H-imidazole-5-carbonyl)piperidin-4-yl]morpholine
N-({3-methyl-7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-2-yl)acetamide
N,1-dimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-indole-2-carboxamide
N-ethyl-4-methyl-5-[3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-thiazol-2-amine
N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
(4aR,7aS)-1-acetyl-4-[2-(2,5-dimethylphenyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(2-methylpropyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1,2-oxazole-3-carboxamide
2-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-5-cyclopropyl-N-methyl-1,2-oxazole-3-carboxamide
3-[2-(methylsulfanyl)pyrimidin-4-yl]-4H-chromen-4-one
N-[(3-fluorophenyl)methyl]-N-[(4-methoxyphenyl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
(2R,6R)-4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(1S,5R)-3-[3-(2-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(benzylsulfamoyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
1-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propan-1-one
4-(6-chloroquinolin-4-yl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(1H-pyrazol-1-yl)-N-[2-(pyridin-2-yl)ethyl]butanamide
{4-[(3-methoxyphenyl)methyl]-1-[2-(3-methylphenyl)benzoyl]piperidin-4-yl}methanol
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
(2S,4R)-N,1-dimethyl-4-[4-(naphthalen-1-yl)-4-oxobutanamido]pyrrolidine-2-carboxamide
methyl 2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]butanoate
N,1,4,6-tetramethyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl[(4-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl][2-(pyridin-2-yl)ethyl]amine
[2-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-1,3-thiazol-4-yl]methanol
1-[7-(1-benzothiophen-3-yl)-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-phenylethan-1-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-ol
methyl 3-[(3S,4R)-1-[(3,4-difluorophenyl)methyl]-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]propanoate
2-(2-cyclopropylacetyl)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-(2-phenylethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{[4-phenyl-5-(1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-{4-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]phenoxy}-N-methylacetamide
1-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-4-phenoxybutan-1-one
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-2-(methylamino)acetamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(3-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-2-(1-methylpiperidin-4-yl)acetamide
(3S,4R)-4-(2-methylphenyl)-1-[4-(1H-pyrazol-4-yl)butanoyl]pyrrolidine-3-carboxylic acid
4-(4H-1,2,4-triazol-3-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}piperidine
{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
N-[(2,4-dimethoxyphenyl)methyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-(2-phenylethyl)thieno[2,3-d]pyrimidine-6-carboxamide
4-{[2-(4-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid