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2-oxo-8-[5-(pyrrolidin-1-yl)pyridazin-3-yl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[4-(benzyloxy)butyl]-6-methylpyrimidin-2-amine
2-methoxy-1-{1-methyl-4-[(2,4,6-trimethylphenyl)methyl]-1,4,9-triazaspiro[5.5]undecan-9-yl}ethan-1-one
N-methyl-N-{2-[(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)amino]ethyl}methanesulfonamide
(4aS,8aS)-2-[1-(4-methylphenyl)piperidin-4-yl]-decahydro-2,7-naphthyridin-4a-ol
1-[3-(benzyloxy)azetidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
N-(3-chloro-4-methoxyphenyl)-3-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-3-yl}propanamide
4-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
1-[4-(1H-pyrazol-3-yl)phenyl]propan-1-ol
6-(2,6-dimethylpyrimidine-4-carbonyl)-3-(4-fluoro-3-methylphenyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-cyclopentanecarbonyl-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
5-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
9-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2,5-difluorobenzoyl)piperidine
1-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-2-(2-methoxynaphthalen-1-yl)-1H-imidazole
1-[3-(2-ethylphenoxy)azetidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
N-[3-(propan-2-yloxy)propyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
N-[(5-methylpyrazin-2-yl)methyl]-2-(1-methylpyrrolidin-2-yl)acetamide
3-(4H-1,2,4-triazol-4-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}benzamide
3-[4-(cyclopentylmethyl)piperazine-1-carbonyl]-4-fluorobenzene-1-sulfonamide
N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)oxolane-2-carboxamide
N,2-dimethyl-3-[(5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-1,3-thiazol-2-yl)amino]benzamide
2-methyl-6-[1-(2-methylphenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]-2,3-dihydropyridazin-3-one
3-(3-chloro-2-methylphenyl)-1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]urea
N-[(2-methylphenyl)(pyridin-4-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
(3S,4R)-1-(dimethyl-1,3-oxazole-5-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-(3-hydroxy-3-phenylpropyl)-N,4-dimethyl-1H-imidazole-5-carboxamide
4-{[3-(trifluoromethyl)phenyl]methyl}piperazine-1-sulfonamide
N-(2,3-dihydro-1H-inden-2-yl)-2,3-dimethylquinoxaline-6-carboxamide
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-[(1-methylpiperidin-4-yl)methyl]piperazine
methyl N-(1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-1-oxopropan-2-yl)carbamate
(4aS,8aS)-2-[4-(pyrrolidin-1-yl)benzoyl]-decahydro-2,7-naphthyridin-4a-ol
N-[(2,3-dimethylphenyl)methyl]-N-methyl-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
N-ethyl-3-methanesulfonyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
1-(4-methoxyphenyl)-2,2-dimethyl-4-(pyrrolidin-3-ylmethyl)piperazine
1-ethyl-3-(piperidine-1-carbonyl)-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
5-methyl-1-(2-oxo-2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
(3R,4S)-4-cyclopropyl-1-(4-methoxy-3,5-dimethylbenzenesulfonyl)pyrrolidin-3-amine
N-[3-(1H-imidazol-1-yl)propyl]-5-methoxy-1-methyl-1H-indole-2-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1,9-dioxaspiro[5.5]undecan-4-amine
4-(1-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-1H-imidazol-2-yl)pyridine
methyl 3-(2,4-dimethylbenzamido)-6-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-2,6-dimethylquinoline-4-carboxamide
3,3-dimethyl-1-({3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}methyl)urea
1-[(2-fluorophenyl)methyl]-3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
N-ethyl-3-(4-hydroxyphenyl)-N-(oxan-4-ylmethyl)-1H-pyrazole-5-carboxamide