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4-chloro-2-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
3-[1-methyl-5-(morpholin-4-yl)-1H-1,2,4-triazol-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
(2S,4R)-4-amino-N-methyl-1-{[4-(prop-2-en-1-yloxy)phenyl]methyl}pyrrolidine-2-carboxamide
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-methyl-3-{[4-(2-methylpropyl)-2-oxopyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
4-(1H-imidazol-2-yl)-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidine
2-methyl-N-{6-methyl-5-[2-(morpholin-4-ylmethyl)phenyl]pyridin-2-yl}propanamide
N-(2-{[3-(dimethylsulfamoyl)-5-{[(4-hydroxy-3,5-dimethylphenyl)methyl]amino}phenyl]formamido}ethyl)acetamide
2,6-dimethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrimidine-4-carboxamide
1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)-2-(4-fluorophenyl)piperidine
3-(3-hydroxy-1,2-oxazol-5-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(4-methyl-1,3-thiazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-benzyl-8-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(3-fluorophenoxy)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxylic acid
N-(1-benzylpyrrolidin-3-yl)-5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-[2-(morpholin-4-ylmethyl)phenyl]-1-[3-(phenylsulfanyl)propyl]urea
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-({[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]amino}methyl)-2,6-dimethylphenyl acetate
methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)[1-(1,3-thiazol-5-yl)ethyl]amine
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3,5-difluoropyridine-2-carboxamide
N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]oxolane-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}ethan-1-one
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-1-hydroxycyclopentane-1-carboxamide
4-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine-3-carbonyl]morpholine
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
1-[2-(dimethylamino)ethyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-oxopyrrolidine-3-carboxamide
2-[(adamantan-1-ylmethyl)({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
N-[4-({[(5-methyl-1,2,4-oxadiazol-3-yl)methyl](propan-2-yl)amino}methyl)phenyl]acetamide
1-[1-(4,6-dimethoxypyrimidin-2-yl)piperidin-4-yl]piperidin-4-ol
1-ethyl-N-[2-(1H-imidazol-1-yl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
2-[1-(3-chloro-4-fluorophenyl)-5-(2-methanesulfonamidoethyl)-1H-1,2,4-triazol-3-yl]acetamide
4-[5-(methoxymethyl)furan-2-carbonyl]-2-[(3-methoxyphenyl)methyl]morpholine
methyl 2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}acetate
3-{[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(pyridin-3-yl)propan-1-one
(3aS,6aS)-2-(ethanesulfonyl)-5-(furan-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(3-methylfuran-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
8-[(2S)-2-amino-2-cyclopropylacetyl]-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-(1H-pyrazol-4-yl)benzamide
[(3S,5R)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]piperidin-3-yl]methanol
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
N-({4-[(3,5-dimethoxyphenyl)methoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
ethyl 4-[({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}carbamoyl)amino]benzoate
6-{4-[(methylsulfanyl)methyl]piperidin-1-yl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
(4aS,8aR)-1-(2-aminoethyl)-6-[3-(thiophen-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
2-{[(4-methoxypyrimidin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide