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3-{2-oxo-2-[4-(9H-purin-6-yl)piperazin-1-yl]ethyl}imidazolidine-2,4-dione
1-ethyl-5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1H-indole
N-[(4-methoxyphenyl)methyl]-2-methyl-N-(pyridin-2-ylmethyl)-1,3-thiazole-4-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]benzamide
2-(4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)phenol
2-(4-fluoro-3-methylbenzenesulfonamido)-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
(2S,4S)-4-amino-1-{[5-(3-chlorophenyl)furan-2-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-(pyrimidin-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(2-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)-1,2,3-thiadiazole-4-carboxamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
4-(2-methylfuran-3-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
9-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(3-methoxypyrazin-2-yl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
methyl (2S,4R)-4-(2-methylquinoline-4-amido)-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidine-2-carboxylate
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-(2-methoxyethyl)piperidine
2-[1-(1H-indol-7-ylmethyl)-3-oxopiperazin-2-yl]-N-methylacetamide
N,N,1-trimethyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
(2S)-2-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carbonyl]pyrrolidine-1-carboxamide
(4aR,7aS)-1-ethyl-4-[2-(pyridin-4-ylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(azepane-1-carbonyl)-N-[2-(methylsulfanyl)ethyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-4-(2-ethylpyrimidin-5-yl)-6-(4-methoxyphenyl)-5-methylpyridine-3-carbonitrile
1-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(pyridin-2-yl)propan-1-one
3-{[1-(quinolin-2-yl)piperidin-4-yl]methyl}benzoic acid
(4aS,8aR)-1-(3-aminopropyl)-6-(quinolin-2-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[2-({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]-N-methylmethanesulfonamide
5-(propan-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
4-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-2-amine
4-[3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]-2-methylbut-3-yn-2-ol
N-[4-(4-{[1-(thiophen-3-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amine
N-[(2-fluorophenyl)methyl]-3-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]propanamide
1-[(1-hydroxycyclohexyl)methyl]-3-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
(3aS,6aR)-5-(isoquinolin-1-yl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-ethyl-1-[(2-fluorophenyl)methyl]-N-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-1-(1,3-benzothiazol-2-yl)piperidin-4-amine
5-chloro-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)pyridine-3-carboxamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(2-hydroxyethyl)-N-methyl-1,3-oxazole-4-carboxamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-methylbutan-1-one
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(3R,4R)-1-(2-chloro-6-fluorobenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
2-[7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-2-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxylic acid
4-(2-methyl-1H-imidazol-1-yl)-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidine-4-carboxylic acid
8-[(3-chlorophenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(3S,4R)-1-benzyl-4-(dimethylamino)piperidin-3-yl]-N-[2-(piperidin-1-yl)ethyl]propanamide
4-{[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylbenzamide
2-{[2-(methoxymethyl)piperidin-1-yl]methyl}-1-methyl-1H-indole
3-[({4-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]-2,2-dimethylpropan-1-ol